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2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-6-methylimidazo[1,2-a]pyridine
1-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-3-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)urea
6-({1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}amino)pyridine-2-carbonitrile
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
4-({3-[2-(trifluoromethoxy)phenyl]-1,2-oxazol-5-yl}methyl)-1,4-oxazepan-6-ol
2-[(1R,3S,3aS,6aR)-5-ethyl-1-(hydroxymethyl)-3-(2-methoxynaphthalen-1-yl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]ethan-1-ol
1-{3-[5-(3,4-dimethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]propyl}-1H-1,2,4-triazole
4-phenyl-3-(piperidin-3-yl)-1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-1-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}urea
N-(1,3-dihydroxypropan-2-yl)-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-[(propan-2-yl)sulfamoyl]-5-(1H-pyrazol-1-yl)benzoic acid
1-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
2-(azepan-1-yl)-1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
N-methyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-phenylethyl)piperidin-3-amine
3-(but-2-yn-1-yl)-5-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
3-{[1-(2-fluoro-6-methoxybenzoyl)piperidin-4-yl]methyl}benzoic acid
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)pyrrolidine-1-sulfonamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-phenoxypiperidine-4-carboxylic acid
(3S)-3-[(6-methoxypyrimidin-4-yl)amino]azepan-2-one
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-3-(2-methoxyphenyl)-N-(oxolan-2-ylmethyl)propanamide
3-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-3,9-diazaspiro[5.5]undecane
2-(3-fluorophenoxymethyl)-4-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,3-oxazole
(3R,4R)-1-(2-chlorobenzoyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-{1-[1-(4-aminopyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
(1R,5R)-6-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(4-fluoro-2-methylbenzenesulfonyl)-2,7-diazaspiro[4.5]decane
4-fluoro-N-(2-{7-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(1H-pyrazol-1-yl)benzamide
3-cyclohexyl-1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]propan-1-one
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-[(4-methylpiperazin-1-yl)sulfonyl]benzamide
(3S,4S)-4-cyclopropyl-1-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
3-(2-methylphenyl)-1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}propan-1-one
N-[(3R,5S)-1-butyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-(5-{[3-(4-chlorophenyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
2-[1-cyclopentyl-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[1-(thiophen-2-yl)ethyl]acetamide
3-benzyl-5-[(4-methanesulfonylphenyl)methyl]-1H-1,2,4-triazole
{3-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-oxopropyl}urea
methyl 3-(1-benzothiophen-2-ylmethyl)-9-[(1-methylpiperidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)-5-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}imidazolidine-2,4-dione
1-[(2-hydroxy-4-methoxyphenyl)methyl]-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
1-(2-methylpyridin-4-yl)-4-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazine
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-[(cyclopropylmethyl)sulfanyl]ethan-1-one
3-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-[2-(diethylamino)ethyl]-1-ethyl-N-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-amino-4-(furan-3-yl)-6-(2-phenylethyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(1S,6R)-9-(5-butylpyridine-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[5-(2H-1,3-benzodioxol-5-ylmethyl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]pyridine
1-{4-[({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]piperidin-1-yl}ethan-1-one
3-{1-[1-(but-3-enoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
1-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one