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2-{2-[1-(1H-pyrazol-3-ylmethyl)piperidin-2-yl]ethyl}pyridine
N-(2-{7-[(4-fluoro-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
5-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
2-[(3R,4S)-3-[(2,5-dimethylpyrimidin-4-yl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]propane-1,3-diol
1-(2-methoxyphenyl)-3-{1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-methyl-5-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)[(4-methylphenyl)methyl]amine
1-[1-(4-methanesulfonylphenyl)ethyl]-2-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-imidazole
3-methyl-1-[3-(thiomorpholine-4-carbonyl)benzenesulfonyl]piperidin-3-ol
1-[2-fluoro-3-(trifluoromethyl)phenyl]-3-[3-(oxolan-3-yl)propyl]urea
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanamide
4-(1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)morpholine
N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(thiophen-2-yl)propanamide
2-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]-2,3-dihydro-1H-isoindole
3,4-dimethyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-5-sulfamoylbenzamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-(4-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}thiophen-2-yl)ethan-1-one
4-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-4-yl]morpholine
(1S,5R)-6-benzyl-3-{[4-(2-hydroxyethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 3-[(3-chlorophenyl)methyl]-1-(4,4,4-trifluorobutanoyl)piperidine-3-carboxylate
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-(pyridin-4-yl)quinoline-4-carboxamide
1-(1-{[1-(4-methoxypyrimidin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]amine
2-methoxy-2-phenyl-N-{1-[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
3-(3-methylbutyl)-8-[2-(2-oxopiperidin-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-fluoro-2-methylphenyl)methyl]acetamide
3-[1-(2,6,8-trimethylquinoline-4-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
2-ethyl-9-[3-(methylsulfanyl)propanoyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-(pyridin-3-yl)acetamide
2-methoxy-N-{1-[1-(3-methoxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
5-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
(1H-imidazol-2-ylmethyl)[(2-methoxyphenyl)methyl](prop-2-en-1-yl)amine
2-{4-[6-(trifluoromethyl)pyridine-3-carbonyl]morpholin-3-yl}acetic acid
3-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridine-2-carbonitrile
3-{[(2-aminopyridin-3-yl)methyl]sulfamoyl}-N-(2-methoxyethyl)-N-methylbenzamide
3-{[(1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)oxy]methyl}pyridine
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-[2-(4-methylphenoxy)ethyl]propanamide
1-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
3-(naphthalene-2-carbonyl)piperidine
N-[1-(2-phenylethyl)piperidin-3-yl]-2-(1H-1,2,4-triazol-3-yl)benzamide
3-(4-chlorophenyl)-4-[(5,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]butanoic acid
methyl 2-{3-[(4-fluorophenyl)amino]piperidine-1-carbonyl}benzoate
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-methoxyfuran-2-carboxamide
2-methyl-N-(oxan-4-yl)thieno[3,2-d]pyrimidin-4-amine
N-{4-[2-(1,2-benzoxazol-3-yl)acetamido]-2-chlorophenyl}propanamide
N-[(4-chlorophenyl)(phenyl)methyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
8-methyl-2-(pyridine-3-sulfonyl)-2,8-diazaspiro[4.5]decane
N-(1,2-oxazol-3-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]benzamide