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N-methyl-2-(naphthalen-2-yloxy)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
2-[4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperazin-1-yl]-4-phenylpyrimidine
4-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)pyrimidine-5-carboxylic acid
{5-fluoro-7-[4-methoxy-3-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
1-cyclopropyl-3-[2-(3-methylpiperidin-1-yl)-2-oxoethyl]-3-(4-phenylphenyl)pyrrolidine-2,5-dione
(1S,5R)-3-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(furan-2-ylmethyl)-N,1-dimethyl-5-({[1-(piperidin-1-yl)cyclohexyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]propanoic acid
N-(1-{1-[(2S)-2-aminobutanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
N,6-dimethyl-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
(1R,3S,5S)-8-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-8-azabicyclo[3.2.1]octan-3-ol
{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}(thiophen-2-yl)methanol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,1-dimethyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N,N-dimethyl-5-{[4-(thian-4-yl)piperazin-1-yl]methyl}pyridin-2-amine
ethyl (4aS,8aR)-6-{pyrazolo[1,5-a]pyridine-3-carbonyl}-decahydro-1,6-naphthyridine-4a-carboxylate
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[(2-methylphenyl)methyl]benzamide
(1S,4S)-2-benzyl-5-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2,5-diazabicyclo[2.2.1]heptane
(3R,4S)-3,4-dimethyl-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperidin-4-ol
3-[(3-phenyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-benzylpiperazine-1-carbonyl)-6-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-6-azaspiro[2.5]octane
2-(methylamino)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)pyridine-4-carboxamide
N-[(4-fluorophenyl)methyl]-1-methyl-5-oxo-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
4-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carbonyl]benzonitrile
4-benzyl-3-(2-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-oxoethyl)piperazin-2-one
N-{1-[1-(2-oxopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
N-cyclopentyl-4-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)benzamide
N-(2-{[5-(2,5-dimethylphenoxymethyl)-1,2-oxazol-3-yl]formamido}ethyl)acetamide
3-{[methyl(prop-2-en-1-yl)amino]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
1-[1'-(2-ethylpyrimidine-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
2-(2,6-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-amino-6-(4-methyl-1,3-thiazol-5-yl)-4-(3-methylthiophen-2-yl)pyridine-3-carbonitrile
2-(3-methyl-1,2,4-oxadiazol-5-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-2-oxo-1,2-dihydroquinazoline-4-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-N-phenyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(4-{[(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amino}piperidin-1-yl)ethan-1-one
(4aS,8aR)-1-(2-methylpropyl)-2-oxo-N-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridine-6-carboxamide
N-(2-methylphenyl)-3-{[(pyridin-3-ylmethyl)carbamoyl]methyl}morpholine-4-carboxamide
2-[(3,4-difluorophenyl)methyl]-8-(1,2-oxazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
(oxolan-2-ylmethyl)(pyridin-4-ylmethyl){[2-(trifluoromethyl)phenyl]methyl}amine
3-{2-[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-1H-imidazol-1-yl}-N,4-dimethylbenzamide
1-(4,6-dimethyl-2-oxo-2H-pyran-5-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N,N-diethyl-6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-{4-chloro-2-[(3-acetamidopiperidin-1-yl)methyl]phenoxy}acetic acid
1-methyl-4-{[1-(2-phenylethyl)-5-(1H-1,2,3,4-tetrazol-1-ylmethyl)-1H-1,2,4-triazol-3-yl]methyl}piperidine
N-(adamantan-2-yl)-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
6-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-N,N,1-trimethyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-(oxan-4-yl)-5-(1,3-thiazol-4-ylmethyl)-1H-1,2,4-triazole
N-methyl-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[(5-methylfuran-2-yl)methyl]acetamide
4-{3-[2-(2,3-difluorophenyl)-1H-imidazol-1-yl]propyl}pyridine