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8-butanoyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-(2-methoxy-4-methylphenyl)-1-(2-methoxyethyl)-4-phenyl-1H-imidazole
1-cyclopentyl-N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)benzamide
1-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}-3-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]urea
1-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)-3-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
3-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyridazine
3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-ol
2-{9-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazine
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylcyclopropane-1-carboxamide
N-ethyl-2-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyrimidin-4-amine
[(4aS,8aR)-6-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-decahydro-1,6-naphthyridin-4a-yl]methanol
3-{[(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
methyl 9-[(4-fluorophenyl)methoxy]-3-[(1-methyl-1H-indol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(4-fluorophenyl)-N-(2-methoxyethyl)-3,5-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
N-({1-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
7-chloro-4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}oxolane-2-carboxamide
(1S,5R)-6-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
N-[4-(1H-pyrazol-1-yl)phenyl]-1-(quinolin-8-ylmethyl)pyrrolidine-2-carboxamide
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl][(3-methylthiophen-2-yl)methyl]amine
N-[(3R,4S)-1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]cyclobutanecarboxamide
1-[(1S,2S)-2-(benzyloxy)cyclohexyl]-3-(1,3-dimethyl-1H-pyrazol-5-yl)urea
methyl 8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
6-(difluoromethyl)-2-[4-({methyl[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
4-[(5,6-dimethylpyridin-3-yl)formamido]-N,4-dimethylpentanamide
N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
5-[1-(2-methoxyethyl)pyrrolidin-3-yl]-1-[4-(methylsulfanyl)phenyl]-1H-1,2,4-triazole
1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-4-(furan-2-carbonyl)-1,4-diazepane
(1S,5R)-3-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(3-fluorophenyl)-3-{1-[1-(3-phenoxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-[1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)pyrrolidin-2-yl]pyridine
3-[2-(dimethylamino)ethyl]-5-[(3-fluorophenyl)methyl]-5-{1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
4'-(2-propoxyethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl 6-{[methyl(thiophen-2-ylmethyl)amino]methyl}-3-[2-(2-methylphenyl)acetamido]thieno[2,3-b]pyridine-2-carboxylate
methyl 2-(5-{1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetate
(3S,5S)-1-[(2-ethylphenyl)methyl]-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
4-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
1-(2-methoxyphenyl)-2,2-dimethyl-4-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperazine
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
2-{1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}-1,3-benzoxazole
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanamide
7-(cyclopropylmethyl)-6-(2-fluoro-4-methoxyphenyl)-N-(2-hydroxypropyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(furan-2-yl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]propanamide
3-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[1-(3-methylpyridin-2-yl)propan-2-yl]benzamide
3-(2-ethylphenoxy)-1-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}azetidine
6-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[3-(furan-2-yl)propyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-[1-(pyrimidin-2-yl)piperidin-3-yl]urea