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2-{4-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(4aR,8aS)-6-[(3,4-difluorophenyl)methyl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
(1R,3S)-7-[4-(1,3-oxazol-5-yl)benzoyl]-7-azaspiro[3.5]nonane-1,3-diol
N-[(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-yl)methyl]acetamide
3-(2,3-dihydro-1H-inden-2-yl)-8-(furan-3-ylmethyl)-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopropyl-5-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-methyl-N-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(2-methyl-1H-indol-1-yl)propan-1-one
N-[2-(diethylamino)ethyl]-N-ethyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
1-{4-[(2-hydroxyethyl)(methyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-4-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-1,2,3-triazole
5-(methoxymethyl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}thiophene-2-carboxamide
4-[2-(3-chlorophenyl)acetyl]-1-(4-methylphenyl)piperazin-2-one
7-[(4-phenylpiperazin-1-yl)methyl]-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1S,5R)-3-(oxan-4-yl)-6-(3-phenyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2S,4S)-4-amino-N,N-diethyl-1-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]pyrrolidine-2-carboxamide
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,3-dimethyl-1H,4H-pyrazolo[3,4-d]imidazole
(2S)-2-(methylamino)-1-[6-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
4-[1-(pyrrolidin-1-yl)ethyl]-1-(thiophen-2-ylmethyl)piperidine
1-{4-[(3-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,2-oxazol-5-yl)methoxy]phenyl}-1H-1,2,4-triazole
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
5-(2-methoxy-4-methylphenoxymethyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
(3R,4R)-1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-4-cyclobutyl-3-methylpiperidin-4-ol
5-propyl-1'-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-N-[3-(methylsulfanyl)propyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
(1S,2S)-2-{4-[2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carbonyl]piperazin-1-yl}cyclohexan-1-ol
2-(3-fluorophenyl)-N-({7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
2-(2H-1,3-benzodioxol-5-ylmethyl)-4-[4-(2-ethylbutyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-(4-{4-chloro-2-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
N-[1-(1H-imidazol-1-yl)butan-2-yl]-2-(morpholin-4-yl)-2-oxoacetamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)but-3-enamide
6,8-dimethyl-3-{1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-imidazol-2-yl}-1,2-dihydroquinolin-2-one
4-[4-(4-propylpyrimidine-5-carbonyl)piperazin-1-yl]quinazoline
N-[(3R,4S)-4-cyclopropyl-1-(2,5-dimethylfuran-3-carbonyl)pyrrolidin-3-yl]-5-methyl-1,2-oxazole-3-carboxamide
2-(cyclopropylamino)-N-(pyridin-3-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
2-hydroxy-N-[(3R,4S)-4-propyl-1-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-3-yl]acetamide
(2S)-N1-[2-chloro-5-(propylcarbamoyl)phenyl]-N2-ethylpyrrolidine-1,2-dicarboxamide
2-{1-[1-(9H-purin-6-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
3-{4-[1-(1H-indol-5-yl)-1H-imidazol-2-yl]phenyl}prop-2-yn-1-ol
N-[(5-fluoro-1H-indol-2-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
1-(4-fluorophenyl)-4-[4-(1H-imidazol-1-yl)benzoyl]-1,4-diazepane
(1S,6R)-N-(3-cyanophenyl)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
2,5-dimethyl-N-[4-(pyrrolidin-1-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-({4-[(2,3-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-3-ethylpiperazin-2-one
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-1,7-dimethyl-2,4-dioxo-1H,2H,3H,4H-pyrido[2,3-d]pyrimidine-5-carboxamide
N-[1-({[2-(4-hydroxyphenyl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
methyl (2S)-4-methyl-2-{3-[5-(phenoxymethyl)-1,3,4-oxadiazol-2-yl]propanamido}pentanoate