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2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxo-N-propylacetamide
1-benzoyl-2-[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidine
5-{1-[5-(2-ethylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(1H-pyrazol-1-yl)propan-2-yl]benzamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]thiophene-2-carboxamide
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)propane-1-sulfonamide
2-(3-{1-[2-(3-fluorophenyl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrazine
N-cyclohexyl-1-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-methyl-N-(oxan-4-yl)benzamide
4-methyl-1-{[4-(propan-2-yl)phenyl]methyl}-1,4-diazepan-5-one
8-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-amino-4-(3,4-dihydroxyphenyl)-6-[3-fluoro-5-(trifluoromethyl)phenyl]pyridine-3-carbonitrile
2-{2-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
8-[(5-ethylpyridin-2-yl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
4-{1,3-dimethyl-4-[3-(propoxymethyl)pyrrolidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]propanamide
1-{4-[(2,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-phenylethan-1-ol
4-{3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
N-[2-(4-fluorophenoxy)ethyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
5-[2-(hydroxymethyl)phenyl]-N-(pyridin-3-yl)furan-2-carboxamide
6-fluoro-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-(1H-1,2,3,4-tetrazol-1-yl)propanamide
2-cyclopentyl-9-(4-fluoro-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-2-{4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}azepane
N-methyl-N-[1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidin-3-yl]acetamide
3-{2-[3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-chloro-N-{[1-(2-ethoxyethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}pyridine-4-carboxamide
3-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-6-(propan-2-yl)-1,2-dihydropyridin-2-one
6-fluoro-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(1-methyl-1H-pyrazol-4-yl)-N-(propan-2-yl)quinoline-4-carboxamide
1-(2-methoxyethyl)-3-(3-methoxyphenyl)-3-{2-oxo-2-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
1-(4-methoxyphenyl)-6,6-dimethyl-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(3-ethyl-1,2-oxazole-5-carbonyl)-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
1-{[5-(4-ethoxyphenyl)furan-2-yl]methyl}-4-(2-methoxyethyl)piperazine
N-[(4-chlorophenyl)methyl]-3-ethyl-3-(hydroxymethyl)piperidine-1-carboxamide
3-[(dimethylamino)methyl]-3-hydroxy-N-(2,4,6-triethylphenyl)piperidine-1-carboxamide
3-(1H-pyrazol-1-ylmethyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]benzamide
4-methoxy-6-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidin-2-amine
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl)(pyrazin-2-ylmethyl)amine
N-(1,3-dihydroxy-2-methylpropan-2-yl)-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(quinoxalin-6-ylmethyl)amine
N-tert-butyl-2-methyl-3-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamido}benzamide
methyl 4-oxo-4-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidin-1-yl}butanoate
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
4-cyclopentyl-N-[2-(1,3-thiazol-2-yl)ethyl]pyrimidin-2-amine
(2E)-4-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]pent-2-enamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[(piperidin-4-yl)sulfamoyl]benzamide
1-{1-[1-(4-chlorophenyl)cyclopropanecarbonyl]piperidin-4-yl}-2-(pyridin-2-yl)-1H-1,3-benzodiazole
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butan-1-one