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3-[2-(2,6-difluorophenyl)ethyl]-1-(furan-2-carbonyl)piperidine
4-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]benzamide
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
N-(2-{[4-(2,2-dimethylpropyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}quinolin-5-yl)acetamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(4-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1,4,6-trimethyl-2-oxo-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-1,2-dihydropyridine-3-carboxamide
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide
(3S,4S)-1-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-4-(propan-2-yloxy)pyrrolidin-3-ol
methyl 2-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]piperidine-1-carboxylate
N-methyl-3-(2-methylpropyl)-N-(pyrazin-2-ylmethyl)-1,2-oxazole-5-carboxamide
5-fluoro-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-methoxybenzamide
N-benzyl-5-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]furan-2-carboxamide
(1S,5R)-3-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(1H-indol-1-yl)propan-2-yl]-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
2-ethyl-N-{[3-(2-methoxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
N-{4-[butyl(methyl)carbamoyl]-2-methylphenyl}furan-2-carboxamide
2-{1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]pyrrolidin-2-yl}pyridine
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)propan-1-one
2-ethyl-9-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-1-{[2-(2-phenylethoxy)phenyl]methyl}pyrrolidine-3-carboxamide
N-benzyl-N-(1,1-dioxo-1λ6-thiolan-3-yl)-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{[4-(2-ethoxyphenyl)piperazin-1-yl]methyl}piperidin-3-ol
1-[3-({[(2,3,6-trifluorophenyl)methyl]amino}methyl)pyridin-2-yl]piperidin-3-ol
N-ethyl-N'-(4-methylphenyl)-N-[3-(morpholin-4-yl)propyl]propanediamide
2-benzyl-N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-1,3-thiazole-4-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
(2H-1,3-benzodioxol-4-ylmethyl)(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
5-(dimethyl-1,2-oxazol-4-yl)-1-phenyl-1H-1,2,4-triazole
methyl 4-({4-[1-(but-2-yn-1-yl)-2,5-dioxo-4-(2-phenylethyl)imidazolidin-4-yl]piperidin-1-yl}methyl)benzoate
1-[(2-fluorophenyl)methyl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
5-[2-(2H-1,3-benzodioxol-5-yloxy)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
4-(1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperazine-2-carbonyl)morpholine
5-(azepane-1-carbonyl)-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
5-(2H-1,3-benzodioxol-5-yl)-1-methyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazole
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl](1,3-thiazol-4-ylmethyl)amine
6-(aminomethyl)-2-[3-({methyl[2-(phenylsulfanyl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N-(1-{[2-(benzyloxy)phenyl]methyl}piperidin-4-yl)methanesulfonamide
6-(3-fluoro-4-methoxybenzoyl)-1-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-fluorophenyl)urea
3-({5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}amino)propane-1,2-diol
N-{3-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindole-2-carbonyl]-4,5-dimethylthiophen-2-yl}-2-methylpropanamide
5-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2,4-diol
N-[2-(cyclohexylsulfanyl)ethyl]-1-(4-hydroxyphenyl)-5-oxopyrrolidine-3-carboxamide
3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-1-(pyrrolidin-1-yl)propan-1-one
4-(4-methyl-1H-pyrazol-1-yl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidine-4-carboxylic acid
1-[(3S)-3-ethylmorpholin-4-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one