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1-(4-methyl-1,3-thiazol-2-yl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
N-[3-(dimethylamino)-1-phenylpropyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
1-{5-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-2-methylphenyl}imidazolidin-2-one
4-{[2-(cyclohexylmethyl)morpholin-4-yl]methyl}-N-methylbenzene-1-sulfonamide
1-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-3-phenylprop-2-yn-1-one
4-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2-(methylsulfanyl)-1,3-thiazole
1-(4-chlorophenyl)-N-{[4-fluoro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutane-1-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-{[4-(1H-imidazol-1-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3-ethoxyphenyl)methyl]-2-(1-methyl-1H-imidazol-2-yl)-N-(prop-2-en-1-yl)benzamide
6-methoxy-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2,3-dihydro-1H-indene-5-carboxamide
N-(4-chlorophenyl)-3-[1-(1,3-thiazole-4-carbonyl)piperidin-3-yl]propanamide
(3aS,6aS)-5-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-(cyclopropylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
6-[1-cyclohexyl-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-2-methyl-2,3-dihydropyridazin-3-one
5-{2-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
2-methyl-6-(2-methylpropyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]pyrimidine-4-carboxamide
1-(3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzoyl)-1,4-diazepane
1-(4-methyl-2-phenylpiperazin-1-yl)-4-(1H-pyrazol-4-yl)butan-1-one
1-[4-({[(4-fluorophenyl)methyl](1-hydroxybutan-2-yl)amino}methyl)phenyl]ethan-1-one
3-[2-fluoro-6-(propan-2-yloxy)phenyl]-6-methylpyridazine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylcyclopentanecarboxamide
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
methyl 6-(3-methylpentanoyl)-2-[(2-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-{4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}-N,N-dimethylacetamide
3-[1-(oxan-4-yl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
ethyl 4-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}piperazine-1-carboxylate
5-oxo-1-[4-(propan-2-yl)phenyl]-N-[3-(pyridin-2-yl)propyl]pyrrolidine-3-carboxamide
1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-[2-(propan-2-yl)phenyl]-2-(trifluoromethyl)morpholine-4-carboxamide
2-tert-butyl-6-(2-chlorobenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-(1H-pyrazol-4-yl)pyridine-3-carboxamide
1-(1-{[4-(benzyloxy)-2-methoxyphenyl]methyl}piperidin-4-yl)ethan-1-ol
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3-benzothiazole-6-carboxamide
(4aS,7aR)-1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2-(benzyloxy)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(2E)-1-{4-[2-(cyclopentylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
4-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
[2-ethoxy-5-({[(3S)-2-oxoazepan-3-yl]amino}methyl)phenyl]methyl acetate
5-[(4-benzylpiperidin-1-yl)methyl]-N-(oxan-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-cyclohexyl-N-(2-hydroxyethyl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(cyclohexylmethyl)-6-oxo-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
1-cyclopentyl-4-[2-(dimethylamino)-2-(3-fluorophenyl)acetyl]piperazin-2-one
3-({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
3-[(4-fluorophenyl)formamido]-N-[1-(1H-pyrazol-1-yl)propan-2-yl]propanamide
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-dimethylpiperidin-3-amine
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2,5-dimethyl-3-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)pyrazine