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N-({5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)pyrrolidine-3-carboxylic acid
N-[(3S,4R)-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
N-(1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
3-[4-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-2,8-diazaspiro[4.5]decane
1-methyl-4-{5-[(5-propylfuran-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}piperazine
5-{1-[(4-fluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
(2S,4S)-N,N-diethyl-4-(furan-2-amido)-1-(3-methylbut-2-en-1-yl)pyrrolidine-2-carboxamide
2-(phenylsulfanyl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-ethyl-8-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-2,6-dimethylquinoline-3-carboxamide
4-{2-[1-(thiophene-2-carbonyl)piperidin-2-yl]ethyl}phenol
1-[(2E)-3-phenylprop-2-en-1-yl]-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
3-(3-fluorophenyl)-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
9-(2-chloro-6-methylbenzenesulfonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
3-[2-(azepan-1-yl)acetamido]-N-(2,5-dimethylphenyl)propanamide
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]methanol
1'-(3-phenyl-1H-pyrazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-amino-2-{4-[(2,6-difluoro-4-methoxyphenyl)methyl]piperazin-1-yl}pyrimidine-5-carbonitrile
N-[(3S)-1-(4-chloro-1H-indole-2-carbonyl)pyrrolidin-3-yl]acetamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(5-fluoro-2-methoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(1H-1,2,4-triazol-1-yl)butanamide
N-cyclohexyl-3-{[6-(propan-2-yl)pyrimidin-4-yl]amino}propanamide
1-(methoxymethyl)-N-[(3R,4S)-4-propyl-1-(pyrazin-2-yl)pyrrolidin-3-yl]cyclobutane-1-carboxamide
(4aR,7aS)-N,N-dimethyl-4-[(6-methylpyridin-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-[3-(4-methoxyphenoxymethyl)piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
1-[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
7-chloro-N-[(3S,4R)-4-ethoxyoxolan-3-yl]-3,5-dimethyl-1-benzofuran-2-carboxamide
2-hydroxy-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-4-(methylsulfanyl)butan-1-one
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-[methyl(1-methylpiperidin-4-yl)amino]ethan-1-one
1-[({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]cyclohexan-1-ol
1-{3-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]phenyl}ethan-1-one
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-(oxolan-3-yl)-5-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]-1,2,4-oxadiazole
N-{1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-yl}acetamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)pyridine-4-carboxamide
ethyl 2-[(5-{4-methyl-12-oxo-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-14-yl}pyrimidin-2-yl)amino]acetate
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-1-(3,4-dimethylpiperazin-1-yl)propan-1-one
4-(1-{[5-(1,2-oxazol-5-yl)thiophen-2-yl]sulfonyl}azetidin-3-yl)pyridine
6-(methylsulfanyl)-2-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
4-ethyl-1-methyl-3-[1-(3-methyl-3-phenylbutanoyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-ethoxyphenyl)-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazine
methyl (2S,4R)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]-4-(naphthalene-1-amido)pyrrolidine-2-carboxylate
3-(2-ethoxyethyl)-2-oxo-1-(prop-2-en-1-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
ethyl 4-benzyl-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-4-carboxylate
1-{[4-(cyclopentyloxy)phenyl]methyl}-4-(pyridin-4-ylmethyl)-1,4-diazepane
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione