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1-(3-chlorophenyl)-4-[1-(3-phenylpropyl)piperidin-3-yl]piperazine
2-chloro-5-{pyrazolo[1,5-a]pyridin-7-yl}benzoic acid
1-[(5-cyclohexylthiophen-2-yl)methyl]-N-methylpiperidine-2-carboxamide
3-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-N-methylpropanamide
2-methyl-4-{3-[3-(morpholin-4-yl)azetidine-1-carbonyl]phenyl}butan-2-ol
N-[(2-chloropyridin-3-yl)methyl]-2-(dimethylamino)-N,4-dimethylpyrimidine-5-carboxamide
methyl 4-(5-{[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N-(1,3-benzothiazol-2-yl)-3-{methyl[1-(1,2-oxazol-3-yl)ethyl]amino}propanamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}pyrrolidin-3-yl]methanol
5,8-dichloro-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
2-methyl-8-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-2,8-diazaspiro[4.5]decane
2-{2-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
2-{4-[(1-methylpiperidin-4-yl)methyl]piperazin-1-yl}-N,N-bis(prop-2-en-1-yl)acetamide
3-(2-methoxyphenyl)-N-[1-({[2-(1,3-thiazol-4-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-methylpiperidine
N'-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N'-(oxolan-2-ylmethyl)butanediamide
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(trifluoromethyl)phenyl]urea
1-[3-(2,3-dihydro-1H-isoindole-2-carbonyl)phenyl]imidazolidin-2-one
3-(2-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
(3R)-3-hydroxy-N-[4-(propylsulfanyl)phenyl]pyrrolidine-1-carboxamide
4-phenyl-1-[6-(pyrimidin-5-yl)pyridine-3-carbonyl]azepane
3-(4-hydroxyphenyl)-N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-2-phenylpropanamide
N-(1-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
(3S,4S)-4-methyl-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine-3,4-diol
2-(3-methoxypropyl)-8-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}propane-1-sulfonamide
3-[(3,4,5-trimethoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[4-(methylsulfanyl)phenyl]-3-(naphthalene-2-carbonyl)piperidine-1-carboxamide
N'1-[2-(2-ethoxyphenoxy)ethyl]-N'1-methylcyclopropane-1,1-dicarboxamide
methyl 3-{[3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
1-(2-methoxyethyl)-5-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[1-(2-amino-6-methylpyrimidin-4-yl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
4-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-1-phenyl-1H-1,2,3-triazole
1-[7-chloro-2-(1H-pyrazol-4-yl)quinoline-4-carbonyl]piperidine-3-carbonitrile
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrazole-3-carboxamide
4-hydroxy-1-{1-methyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carbonyl}piperidine-4-carboxylic acid
N-methyl-N-[2-(morpholin-4-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
3-({4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepan-1-yl}methyl)-6-methyl-1,2-dihydroquinolin-2-one
5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-N-(pyridin-4-ylmethyl)pyridin-2-amine
7-(cyclopropylmethyl)-2-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-2,7-diazaspiro[4.5]decane
2-amino-4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
6-{[4-(azocane-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
1-ethyl-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-(thiophen-3-ylmethyl)piperidine
4-(1-ethyl-1H-imidazol-2-yl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
(4aR,7aS)-1-(2-methoxyethyl)-4-[(4-oxo-4H-chromen-3-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(2S)-1-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
2-amino-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)-4-(pyridin-4-yl)pyridine-3-carbonitrile
4-(1H-imidazol-1-yl)-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)benzamide