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3-(3-hydroxyquinoxalin-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]propanamide
1'-(dimethyl-1,2-oxazole-4-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N,3-dimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-4-oxo-3,4-dihydroquinazoline-7-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-2,8-diazaspiro[4.5]decane-2-carboxamide
9-(2-methoxyethyl)-1-methyl-4-[2-oxo-2-(piperidin-1-yl)ethyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{imidazo[1,2-a]pyrimidin-6-ylmethyl}-3-(4-methylphenoxymethyl)piperidine
1-[(2-methylphenyl)methyl]-N-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-cyclopropyl-N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,2-oxazole-3-carboxamide
2-({[(1R,2R,3S,4S)-3-aminobicyclo[2.2.1]heptan-2-yl]formamido}methyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(4S)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
N-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
[3-(dimethoxy-1,3,5-triazin-2-yl)phenyl]methanol
2-[2-(1,2,3,4-tetrahydroisoquinolin-5-yl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
2,4-dimethyl-5-{[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,3-thiazole
1-(2-methanesulfonylethyl)-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
3-benzyl-1-[(4-fluorophenyl)methyl]-6-(thiolan-3-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)benzamide
9-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
(2S,4R)-4-amino-N-ethyl-1-{1H,3H,4H,5H-thiopyrano[4,3-b]indole-8-carbonyl}pyrrolidine-2-carboxamide
N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}oxolane-3-carboxamide
1-(4-fluorophenyl)-4-[3-(phenylamino)piperidin-1-yl]butane-1,4-dione
N-(2,3-dihydro-1H-inden-2-yl)-3-(2-oxoimidazolidin-1-yl)-N-propylbenzamide
7-(propan-2-yl)-2-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
4-(7-fluoro-2-methylquinoline-4-carbonyl)-7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
4-(3-methylphenyl)-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4H-1,2,4-triazole
5-{2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[2-(dimethylamino)-4-{[1-(4-methylpyridin-2-yl)propyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
(2S)-2-[(1-cyclobutanecarbonylpiperidin-4-yl)formamido]-3-phenylpropanamide
(2S,4R)-4-amino-N-(propan-2-yl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]pyrrolidine-2-carboxamide
dimethyl({[(3S,4R)-1-[(2E)-3-phenylprop-2-en-1-yl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
N-[(3R,4S)-1-cyclopentyl-4-(3-methoxyphenyl)pyrrolidin-3-yl]-2-methoxyacetamide
(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[3-(1,3-thiazol-4-yl)phenyl]pyrrolidine-1-carboxamide
3-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-1-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
1-[7-(5,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
2-(adamantan-1-yl)-N-cyclopentylacetamide
({5-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N'-(3,5-dimethylphenyl)-N-(3-propoxypropyl)propanediamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}acetamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-fluoro-3-hydroxy-N-methylbenzamide
methyl 3-(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)propanoate
7-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
(2S)-2-amino-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-4-hydroxybutanamide
1-[(4-methoxyphenyl)methyl]-3-({[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}methyl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
2-{4-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]piperidin-1-yl}acetamide
(3aR,7aS)-2-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-(3-hydroxy-3-methylbutyl)-N-[1-(5-methylpyridin-2-yl)ethyl]benzamide
N-[(3-methylpyridin-2-yl)methyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
1-[4-(4-methoxy-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenoxy)piperidin-1-yl]ethan-1-one