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2,6-dimethoxy-N-[1-(2-phenylethyl)piperidin-3-yl]pyridine-3-carboxamide
N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]-4-(2-oxopyrrolidin-1-yl)benzamide
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-(1-{1-[2-(oxolan-3-yl)ethyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
4-{[5-(pyridin-2-yl)thiophen-2-yl]sulfonyl}morpholine-2-carboxylic acid
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine
3-chloro-N-cyclopentyl-4-[(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]benzamide
2-{[(3R,5S)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1-[(4-methoxynaphthalen-1-yl)methyl]pyrrolidin-3-yl]sulfanyl}-1H-1,3-benzodiazole
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-oxopyrrolidin-1-yl)benzamide
(2S,4S)-1-benzyl-N-ethyl-4-[2-(pyridin-2-yl)acetamido]pyrrolidine-2-carboxamide
9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-amino-1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}hexan-1-one
1-{4-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]phenyl}imidazolidine-2,4-dione
2-ethyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(1-{[3-(cyclopentyloxy)phenyl]methyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
N,N-dimethyl-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
2-butyl-8-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-benzyl-1-(2-ethoxyethyl)-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
methyl 6-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]carbamoyl}amino)-1,2,3,4-tetrahydroquinoline-1-carboxylate
(1S,6R)-3-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(3S,4R)-1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-4-phenylpyrrolidine-3-carboxylic acid
9-[2-hydroxy-4-(methylsulfanyl)butanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-1-methylpiperidine-3-carboxamide
N-cyclohexyl-5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
[1-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)piperidin-4-yl](thiophen-2-yl)methanol
N5-(1,3-benzoxazol-2-ylmethyl)-N5,N6,N6-trimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-cycloheptyl-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N,2-dimethyl-4-oxo-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
N-cyclopropyl-4-methoxy-2-{[1-(1,3-oxazole-5-carbonyl)piperidin-4-yl]oxy}benzamide
1-[(2-ethylpyrimidin-4-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
1-(pyridin-3-ylmethyl)-4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine
2-{1-[(4-ethylphenyl)methyl]-5-{imidazo[1,2-a]pyrimidin-2-yl}-1H-1,2,4-triazol-3-yl}acetamide
N'-[3-(cyclohexyloxy)-2-hydroxypropyl]-N-(2-fluoro-5-methylphenyl)butanediamide
3-methyl-12-(3-methylphenyl)-1,2,4,5,10,11-hexaazatricyclo[7.3.0.02,6]dodeca-3,5,7,9,11-pentaene
1-[(1S)-1-[1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]ethyl]-1H-1,2,3,4-tetrazole
10-methoxy-5-[(6-methoxypyridin-3-yl)methyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
ethyl 3-{[5-(cyclooctylcarbamoyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridin-3-yl]formamido}propanoate
1-(6-cyanopyridin-3-yl)-3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]urea
2-phenoxy-N-[2-(7-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
5-ethyl-5-[1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
1-[(2E)-but-2-en-1-yl]-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,4-diazepan-6-ol
3-(aminomethyl)-4-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]but-2-yn-1-one
N-methyl-3-(6-oxo-1,6-dihydropyridazin-3-yl)-N-[(4-phenoxyphenyl)methyl]propanamide
2-(5-{[4-(pyrrolidin-1-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
1-[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-(furan-2-carbonyl)-1,4-diazepane
3-(2-chlorophenyl)-5-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,2-oxazole-4-carboxamide
N-cyclohexyl-N-(prop-2-yn-1-yl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3-ethyl-1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]piperidine-3-carboxylic acid