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1-(2-methoxypyridine-4-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-{[3-(methylsulfanyl)phenyl]methyl}urea
N6-cyclopentyl-N5-methyl-N5-(1,3-thiazol-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-[2-(dimethylamino)ethyl]-3-ethyl-1-(3-fluoro-5-methylphenyl)urea
4-[4-(1H-imidazol-2-yl)piperidin-1-yl]-5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidine
5,6-dimethyl-N4-(2-propoxypropyl)pyrimidine-2,4-diamine
(3S,4R)-3-ethyl-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-methylpiperidin-4-ol
N-({7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,5-dimethylfuran-3-carboxamide
2-(dimethylamino)-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-(2-methylphenyl)pyridine-3-carboxamide
3-[2-(2,3-difluorophenyl)acetyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-3-yl]methanol
8-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
N-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carboxamide
2-methyl-N-[4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-4,5,6,7-tetrahydro-1,3-benzothiazol-4-amine
4-[4-(4-methylphenoxy)piperidine-1-carbonyl]-1λ6-thiane-1,1-dione
7-(2,2-dimethylpropyl)-2-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
(1S,5R)-3-benzyl-6-(pyridine-3-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
N-(2-{[2-(2-aminoethyl)quinazolin-4-yl]amino}ethyl)-N-methylmethanesulfonamide
5-fluoro-2-{1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-4-yl}-1H-1,3-benzodiazole
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[4-(1H-pyrazol-1-yl)butan-2-yl]acetamide
N-[2-(2-fluorophenyl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]amine
N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2,3-dihydro-1-benzofuran-2-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-[4-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)phenyl]acetamide
1-{3-[4-({[(3,4-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
1-ethyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-(1-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N,1,3,6-tetramethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-[(3-methoxyphenyl)methyl]-2-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
3-methyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
6-(hydroxymethyl)-N-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]-1,4-oxazepane-4-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-fluoro-4-hydroxy-N-(2-methoxyethyl)quinoline-3-carboxamide
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-4-(pyridin-2-ylmethyl)piperazine
N-[3-({[(3,4-difluorophenyl)methyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
N'-cycloheptyl-N-ethyl-N-(oxolan-2-ylmethyl)butanediamide
2,2-dimethyl-6-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-3,4-dihydro-2H-pyran-4-one
4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-1-(thiophen-2-ylmethyl)piperidine
1-(1-ethyl-1H-pyrazole-5-carbonyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
N-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
1-cyclohexyl-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)piperidine-4-carboxamide
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
N1-(4-methylpyridin-2-yl)-N2-[2-(morpholine-4-carbonyl)pyridin-4-yl]ethane-1,2-diamine
2-methyl-6-(propan-2-yl)-N-[1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-4-amine
7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-2-(pyridine-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
1-[benzyl(methyl)amino]-3-{5-[(cyclobutylamino)methyl]-2-methoxyphenoxy}propan-2-ol
(2E)-1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}-3-(pyridin-4-yl)prop-2-en-1-one