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5-(2-methoxyphenoxymethyl)-N-(1-phenylcyclopropyl)-1H-pyrazole-3-carboxamide
3-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}benzonitrile
3-(1H-imidazol-2-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
1-ethyl-4-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}piperidine
N-[(5-methylthiophen-2-yl)methyl]-5-oxo-1-(propan-2-yl)-N-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
3-(3-methoxypropyl)-1-(trimethylpyrimidin-4-yl)piperidine-3-carboxylic acid
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}oxane-4-carboxamide
4-[({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)methyl]-1-methylpiperidin-4-ol
6-{1-cyclohexyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
1-cyclohexyl-4-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}piperidine
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[(3E)-4-methylhex-3-en-1-yl]piperidine
2-[({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]-6-ethoxyphenol
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxamide
3-(2-chloro-4-methylphenyl)-1-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}urea
4-(5-chloropyridin-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
6-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-3-phenylpyrazolo[1,5-a]pyrimidine
1-benzyl-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N,2-dimethyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carboxamide
5-{3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanoyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-amino-6-(1H-pyrrol-2-yl)-4-[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]pyridine-3-carbonitrile
2-(3-{3-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]phenyl}-1H-pyrazol-1-yl)acetamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-(2-methylbut-3-yn-2-yl)acetamide
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)benzamide
3-methyl-5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)cinnoline
N-(2-fluorophenyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carboxamide
4-{4-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]phenyl}-4H-1,2,4-triazole
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-1-methyl-5-phenyl-1H-pyrazole-3-carboxamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-(6-methoxypyridin-2-yl)-2-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenol
3-(5-methylfuran-2-yl)-N-(5-oxo-1-phenylpyrrolidin-3-yl)-1H-pyrazole-5-carboxamide
2-cyclopropanecarbonyl-8-(2,4-dimethylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
5-ethyl-N,2,3-trimethyl-N-(1,2-oxazol-5-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
methyl (2S)-1-[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carbonyl]pyrrolidine-2-carboxylate
1-(3-{[(butan-2-yl)(pyridin-3-ylmethyl)amino]methyl}-1H-indol-1-yl)ethan-1-one
5-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(naphthalen-1-ylmethyl)-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(benzylsulfamoyl)({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amine
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
2-methyl-9-(1-methyl-1H-pyrrole-2-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(2S)-2-amino-N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-3-(1H-imidazol-4-yl)propanamide
1-cyclohexyl-3-{2-[(3R)-3-hydroxypyrrolidin-1-yl]-2-oxoethyl}-2,6,6-trimethyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-[(1R,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetic acid
5-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
(3S)-1,3-dimethyl-4-{3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanoyl}piperazin-2-one
1-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
3-phenyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
5-(2-methoxyphenoxymethyl)-N-[(4-methylphenyl)methyl]-1H-pyrazole-3-carboxamide
2,2-dimethyl-N-{5-methyl-3-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]thiophen-2-yl}propanamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(pyrimidin-2-yl)piperidin-3-yl]propanoic acid