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N-(3-methyl-4-pentanamidophenyl)-1H-imidazole-2-carboxamide
7-methyl-2-[3-(2-oxopyrrolidin-1-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
9-(cyclopropylmethyl)-1-methyl-4-(6-methylpyrimidin-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
N-(2-methoxyethyl)-1-[1-(2-methylbenzoyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
3-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetamido]-N-cyclohexyl-2-methylbenzamide
3-{2-oxo-2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethyl}imidazolidine-2,4-dione
methyl 6-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyrazine-2-carboxylate
3-[(3-methoxyphenyl)methyl]-7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecane
methyl 4-({[1-(carbamoylmethyl)piperidin-4-yl]carbamoyl}amino)-2-chlorobenzoate
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
(3S,4S)-4-[(1H-imidazol-2-ylmethyl)(methyl)amino]-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-ol
methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
5-cyclobutanecarbonyl-1'-(1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-(4-acetylphenoxymethyl)-N-[2-(3-hydroxypiperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
N-(1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N,2-dimethylfuran-3-carboxamide
N-tert-butyl-2-(6-methoxy-4-methylpyridin-3-yl)benzene-1-sulfonamide
1-[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
1-(5-{[4-(dimethylamino)piperidin-1-yl]methyl}-2-methoxyphenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
5-[(2-chloro-4-fluorophenyl)methyl]-1-methyl-3-(propan-2-yl)-1H-1,2,4-triazole
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
N-(3,4-dimethoxyphenyl)-4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
4-[(2,4-dimethoxyphenyl)methyl]-7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]benzonitrile
N'-cyclopentyl-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]butanediamide
(4aS,8aR)-6-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-{[({2-[(2-chlorophenyl)methoxy]-6-methylquinolin-3-yl}methyl)amino]methyl}-1λ6-thiolane-1,1-dione
N-[(3R,4S)-4-cyclopropyl-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidin-3-yl]methanesulfonamide
N-methyl-3-{methyl[(2,4,5-trimethylphenyl)methyl]amino}butanamide
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
N-[2-(dimethylsulfamoyl)ethyl]quinoxaline-5-carboxamide
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)(3-methylbut-2-en-1-yl)amine
(2R,6R)-11-methoxy-4-{[(2-methylbutan-2-yl)carbamoyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(2E)-N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-3-(thiophen-2-yl)prop-2-enamide
N-(cyclohex-1-en-1-ylmethyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
4-(3-hydroxy-4-methylbenzoyl)-1-(2-methoxyphenyl)piperazin-2-one
3-(3-methoxyphenyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
1-(cycloheptylmethyl)-4-(2-methoxyethoxy)piperidine
1-(cyclopropylmethyl)-4-[2-(3-methoxyphenyl)ethyl]piperazine
3-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(1H-1,2,4-triazol-1-yl)ethyl]propanamide
N-(3-{2-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-3-oxopropyl)acetamide
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(4-methoxyphenyl)methyl]piperidine
5-(4-fluorophenyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(methoxymethyl)-1H-pyrazole-4-carbonyl)-4-propylpiperazine
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1,4,6-trimethyl-3-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one