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2-(5-{thieno[2,3-d]pyrimidin-4-yl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
1-{[3-(5-methylfuran-2-yl)phenyl]methyl}-4-(oxolane-2-carbonyl)-1,4-diazepane
[(3R,4S)-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-(1-benzofuran-5-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-cycloheptanecarbonyl-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(3-methoxyphenyl)ethyl]methylamine
4-(2,3-dihydro-1H-inden-5-yloxy)-1-(1H-pyrazole-3-carbonyl)piperidine-4-carboxylic acid
3-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}-N-(oxolan-3-yl)benzene-1-sulfonamide
4-ethyl-3-{1-[2-(ethylamino)-5-methylbenzoyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-hydroxyethyl)-N-(4-phenylbutan-2-yl)-1H-1,3-benzodiazole-5-carboxamide
(1S,5R)-6-[(3-fluoro-2-methylphenyl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
1-[4-({[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}amino)piperidin-1-yl]ethan-1-one
2-fluoro-N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)-5-sulfamoylbenzamide
2-(phenoxymethyl)-5-(3-propoxypiperidine-1-carbonyl)pyrimidin-4-ol
2-[2-(3-methylpiperazin-1-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]isoquinoline-3-carboxamide
3-(4-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(2-methylphenyl)-1,4-diazepane
methyl 2-[8-(1-benzofuran-2-ylmethyl)-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
(3S,4S)-3-hydroxy-4-{methyl[2-methyl-2-(morpholin-4-yl)propyl]amino}-1λ6-thiolane-1,1-dione
(4S)-4-(methoxymethyl)-1-(4-methoxyquinoline-2-carbonyl)-3,3-dimethylpiperidin-4-ol
2-(dimethylamino)-2-(3-fluorophenyl)-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-{spiro[2.5]octan-1-ylmethyl}propanamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methoxyethoxy)ethan-1-one
3-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
N-[3-({[3-(pyrrolidin-1-yl)propyl]carbamoyl}methoxy)phenyl]propanamide
(3aR,6aS)-2-[(3-chloro-4-fluorophenyl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole
2-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidin-2-yl}pyridine
4-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}-2-methylphenol
1-[4-(2-chlorophenoxy)piperidin-1-yl]-3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropan-1-one
2-[(2-methyl-1,3-oxazol-4-yl)methyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
N-[2-(2-chlorophenoxy)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
3-{5-amino-6-[4-(ethanesulfonyl)piperazin-1-yl]pyrazin-2-yl}phenol
8-methoxy-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(4-{4-[(4-{[2-(2-methoxyphenyl)ethyl]amino}quinazolin-2-yl)methyl]piperazin-1-yl}phenyl)ethan-1-one
2-{[(3S,4R)-4-ethoxyoxolan-3-yl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-{1-[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]piperidin-3-yl}-3-phenylpropan-1-one
5-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-amine
7-(propan-2-yl)-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)piperidin-4-ol
2-({2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl}amino)-N-(pyrazin-2-yl)acetamide
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(furan-2-ylmethyl)benzamide
3-[2-({2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,3-oxazolidin-2-one
2-(4-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrimidine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
2-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
methyl 5-{[(2,4-dimethylphenyl)methyl]amino}-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide