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3-(pyrrolidine-1-sulfonyl)-5-(quinolin-5-yl)benzoic acid
5,7-dimethyl-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
8-[2-(3,4-dichlorophenoxy)acetyl]-2-methyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-{1-[(5-methylfuran-2-yl)methyl]-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-methyl-N-(1-methylpiperidin-4-yl)-3-[1-(3-phenylprop-2-ynoyl)piperidin-3-yl]propanamide
1-(3-aminoazepan-1-yl)-3-(3-chloro-1H-1,2,4-triazol-5-yl)propan-1-one
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-4-methylphenyl)urea
1-[(2,6-difluorophenyl)methyl]-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(1,3-benzothiazol-2-yl)ethyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(furan-2-ylmethyl)-5-(oxolan-2-yl)thiophene-2-carboxamide
1-(4-ethylpiperazin-1-yl)-3-[3-({methyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-(2H-1,3-benzodioxol-5-yl)-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
4-benzyl-3-ethyl-N-(furan-2-ylmethyl)-5-oxo-1,4-diazepane-1-carboxamide
2-(ethylamino)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidine-5-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-oxo-1,3-oxazolidine-4-carboxamide
1-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
(1S,5R)-3-(4-chloro-2-hydroxybenzoyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{5-[(benzylamino)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
1-(1-benzoxepine-4-carbonyl)-3-(2-fluorophenyl)pyrrolidine
3-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
4-chloro-N-[1-(methoxymethyl)cyclopentyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
3-{4-[2-(3-methoxyphenyl)-1,3-benzoxazole-6-carbonyl]piperazin-1-yl}propanamide
3-[5-(cyclohex-3-en-1-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
5-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-5-(morpholine-4-carbonyl)pyridin-2-amine
1-ethyl-4-{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperazin-2-one
2-methyl-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-4-carboxamide
2-(4-tert-butylphenoxymethyl)-4-hydroxy-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrimidine-5-carboxamide
2-[8-benzyl-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxyethan-1-one
5-(3-chlorophenyl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1,2,4-triazin-3-amine
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
3-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide
1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxypropyl)piperidine
(1S,9R)-11-(3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2-(pyridin-2-ylsulfanyl)acetamide
(3R,4R)-1-[3-(1H-imidazol-2-yl)benzoyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-(3-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-3-oxopropyl)acetamide
2-[({4-[3-(azepan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)(methyl)amino]-N-methylacetamide
8-(3,5-difluoropyridine-2-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
3-[(dimethylamino)methyl]-1-[2-(pyridin-3-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-3-ol
1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
1-(6-chloro-2-methylpyridin-3-yl)-3-[1-(2,4-dimethoxyphenyl)ethyl]-3-methylurea
4,4,4-trifluoro-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazole