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1-[2-(4-methoxy-4-phenylpiperidin-1-yl)-2-oxoethyl]-5-methylpyrrolidin-2-one
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}oxy)benzamide
4-ethyl-1-{2-oxo-2-[2-(thiophen-2-yl)azetidin-1-yl]ethyl}-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]benzenesulfonamide
2-methyl-3-{2-oxa-7-azaspiro[4.5]decane-7-carbonyl}-4,5,6,7-tetrahydro-1-benzofuran-4-one
1-(oxolane-2-carbonyl)-4-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}piperazine
methyl 7-oxo-3-(3-phenylpropyl)-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[(furan-2-ylmethyl)amino]-5-methyl-N-(3-methylbutyl)thieno[2,3-d]pyrimidine-6-carboxamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(1H-imidazol-1-yl)propan-1-one
(6R)-6-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,3-diazinane-2,4-dione
2-(2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
3-[({2-[(2-methylphenyl)amino]-1,3-thiazol-5-yl}methyl)(prop-2-en-1-yl)amino]-1λ6-thiolane-1,1-dione
N-(1-benzylpyrrolidin-3-yl)-3-[1-(1,2,3-thiadiazole-4-carbonyl)piperidin-4-yl]propanamide
2-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-2-yl}-1H-1,3-benzodiazole
methyl (2S)-2-{[5-amino-2-ethyl-1-(3-methoxypropyl)-1H-1,3-benzodiazol-7-yl]formamido}-3-methylbutanoate
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
4-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methoxy}benzamide
2-(1H-1,3-benzodiazol-1-yl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}propanamide
N-methyl-N-(2-phenyl-1-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}ethyl)pyridine-2-carboxamide
5-fluoro-2-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]piperidin-2-yl}-1H-1,3-benzodiazole
2-(cyclopropylmethyl)-8-(4,4,4-trifluorobutanoyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]quinoxaline
5-(6-chloroquinolin-2-yl)-N,N-dimethylthiophene-2-carboxamide
3-(2,5-dimethylphenyl)-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-pyrazole
1-{1-[2-(prop-2-en-1-yloxy)benzoyl]piperidin-4-yl}pyrrolidin-2-one
4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)-N,N-dimethylpiperidine-1-sulfonamide
6-methoxy-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[2-(3-methoxyphenyl)piperidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
1-(4-methoxyphenyl)-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]piperidin-4-amine
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(pyridin-2-yl)ethyl]propanamide
N-{2-[5-(3,4-difluorophenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}methanesulfonamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1H-1,2,3-benzotriazole-5-carboxamide
5-methyl-N-(3-phenoxypropyl)pyrazolo[1,5-a]pyrimidin-7-amine
(1S,5R)-6-methyl-3-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{2-[1-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1H-imidazol-4-yl]ethyl}acetamide
1-(2-methyl-6-propylpyrimidin-4-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]piperidin-4-amine
2-[benzyl({[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
4-(3-methylphenoxy)-1-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperidine-4-carboxylic acid
2-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)-4-(pyridin-2-yl)phenol
4-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridine
3-cyclopropyl-1-phenyl-5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepin-9-yl}-1H-1,2,4-triazole
N-(4-{[(3S,4S)-3,4-dihydroxypiperidin-1-yl]sulfonyl}phenyl)acetamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)hexanamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-[2-(3-methylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(4-chlorophenyl)-N-{[1-(thiophene-3-carbonyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
1-(furan-2-ylmethyl)-N-[2-(pyridin-3-yl)ethyl]piperidine-3-carboxamide
1-[1-(2-methylbenzoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
benzyl N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}carbamate
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
2-methyl-6-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one