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N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
1-[(4-fluorophenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)-1-[(1-phenylcyclopentyl)methyl]pyrrolidin-2-one
methyl 5-{[(2-fluoro-5-methoxyphenyl)methyl]amino}-3-(furan-2-amido)-1-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[(5-methylthiophen-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
2-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(4-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenyl)imidazolidin-2-one
1-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-3-(morpholin-4-yl)propan-1-one
(2S,4S)-4-[4-(4-chlorophenyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxylic acid
8-chloro-N-(2-methoxyethyl)-2-methyl-N-(thiophen-3-ylmethyl)quinoline-4-carboxamide
5-[(2-chlorophenyl)methyl]-5-[1-(3,4-dimethoxybenzoyl)piperidin-4-yl]imidazolidine-2,4-dione
2-methyl-6-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
3-chloro-N-[3-(1H-imidazol-1-yl)propyl]-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
2-benzyl-8-(morpholine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-methyl-N-(oxan-2-ylmethyl)-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
N-[(3-hydroxyphenyl)methyl]-N-methyl-3-(piperidin-3-yl)benzamide
(3R,5R)-5-(pyrrolidine-1-carbonyl)-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-3-carboxamide
7-(1-aminocyclobutanecarbonyl)-N4-(2-ethoxyethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(2S,4R)-4-(2-cyclopentylacetamido)-N-ethyl-1-(5-methyl-1,2-oxazole-3-carbonyl)pyrrolidine-2-carboxamide
N-(furan-3-ylmethyl)-1-(pyrimidin-2-yl)piperidin-3-amine
(1S,5R)-6-(cyclopropylmethyl)-3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3-hydroxypropyl)-8-[3-(1H-pyrrol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
2-({[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]amino}methyl)-8-fluoroquinolin-4-ol
6,7-dimethyl-4-[({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)methyl]-2H-chromen-2-one
N-methyl-1-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperidin-4-amine
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-{[3-(trifluoromethyl)phenyl]methyl}urea
6-[(4aS,8aR)-1-(3-methoxypropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]pyridine-3-carboxamide
3-(1-tert-butyl-4-phenyl-1H-pyrazol-5-yl)-1-methyl-1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]urea
2-[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
N-(1-benzyl-5-oxopyrrolidin-3-yl)-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
7-[(3E)-4-phenylbut-3-enoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
(2S,4R)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-[(4-fluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)(propyl)(pyridin-3-ylmethyl)amine
methyl (2R,4S)-4-hydroxy-1-(4-methoxy-3-methylbenzoyl)piperidine-2-carboxylate
4-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline
5-[(methylsulfanyl)methyl]-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)furan-2-carboxamide
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
1-{[1-(propan-2-yl)piperidin-4-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
N-[2-phenyl-2-(piperidin-1-yl)ethyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
dimethyl[1-(4-{[(1R,5S,6S)-6-(pyrrolidine-1-carbonyl)-3-azabicyclo[3.1.0]hexan-3-yl]methyl}phenyl)ethyl]amine
3-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-methyl-1-(3-phenylphenyl)urea
2-(2-chloro-4-fluorophenyl)-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
(1R,3S)-3-(2-hydroxyethoxy)-7-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-7-azaspiro[3.5]nonan-1-ol
(4aS,7aR)-1-(2-chloro-5-fluorobenzoyl)-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2,4,5-trimethylbenzamide
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}[(5-methoxy-1H-indol-2-yl)methyl]amine
2-[4-(benzyloxy)piperidin-1-yl]-4-(pyrrolidine-1-carbonyl)pyridine
(2S)-4-methyl-2-phenyl-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperazine