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N-{4-[4-({[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}amino)piperidin-1-yl]phenyl}cyclopentanecarboxamide
2-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(2S)-N-[(3-chlorophenyl)methyl]-2-acetamido-3-(1H-imidazol-4-yl)-N-propylpropanamide
2-{1-[2-(1H-imidazol-5-yl)ethyl]-1H-pyrazol-4-yl}-N,N,7,8-tetramethylquinoline-4-carboxamide
2-[4-(1,3-oxazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(oxan-4-yl)benzamide
(3S,4R)-4-(3-methoxyphenyl)-1-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}pyrrolidine-3-carboxylic acid
2-(3-methoxyphenoxymethyl)-N-methyl-N-(2-methylpropyl)-1,3-oxazole-4-carboxamide
4-[1-(1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)ethyl]morpholine
1-{1-[(4-ethynylphenyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-(5-chlorothiophen-2-yl)-1-[(1-propyl-1H-pyrazol-4-yl)methyl]-1H-imidazole
N-cyclohexyl-N-[(4-fluorophenyl)methyl]morpholine-2-carboxamide
(3S,7S)-5-(1-methyl-1H-pyrrole-2-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl){[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}amine
1-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-hydroxyphenyl)ethan-1-one
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-propylpiperazine
1-[1-(4-chlorophenyl)cyclopropanecarbonyl]-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
2-benzyl-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,3-benzoxazole
4-[(8-chloroquinolin-2-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
4-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
1-(2-methyl-1-benzofuran-7-carbonyl)-4-(piperidine-1-carbonyl)piperidine
2-methyl-5-[1-(propan-2-yl)-1H-imidazol-2-yl]quinoline
1-[(4-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}phenyl)methyl]pyrrolidine
1-{1-[(6-methoxy-2H-chromen-3-yl)methyl]piperidin-3-yl}-4-phenylpiperazine
1-(benzenesulfonyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpiperidin-3-amine
3,5-dimethyl-4-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2-oxazole
5-methoxy-2-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4H-pyran-4-one
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(3,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-4-fluorobenzamide
1-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3-(propan-2-yl)urea
9-(2-ethyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-amino-1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-N-methylpyrrolidine-2-carboxamide
N,N-dimethyl-5-{1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H-imidazol-2-yl}pyrimidin-2-amine
4-chloro-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
3-({5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}amino)propane-1,2-diol
N-(2,3-dimethylphenyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
3-benzyl-1-(3-methoxypropyl)-8-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2E)-3-(4-methoxyphenyl)-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)prop-2-enamide
{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(quinoxalin-6-ylmethyl)amine
N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]-4-phenylbutanamide
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N,5,6-trimethylthieno[2,3-d]pyrimidin-4-amine
2-methyl-4-(4-{[1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]methyl}phenyl)but-3-yn-2-ol
N-benzyl-1-{2-[3-(4-methoxyphenyl)propanamido]ethyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
5-(3-propyl-1,2,4-oxadiazol-5-yl)-2-(pyridin-4-yl)pyrimidine
4-(2-methoxyethoxy)-1-[(5-phenylthiophen-2-yl)methyl]piperidine
2-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-[2-(1-methylpiperidin-3-yl)ethyl]acetamide
4-(2,5-dimethoxyphenyl)-3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4H-1,2,4-triazole
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethane-1,2-dione
2-cyclohexyl-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)acetamide