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N-(adamantan-1-yl)-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methylbenzamide
N'1-[(3R,4S)-1-(4-methylpent-3-en-1-yl)-4-propylpyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
3-[2-(5-methyl-2-oxo-5-phenylpiperidin-1-yl)ethyl]-1,3-oxazinan-2-one
5-(piperidin-1-yl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[1-(3-methylpyridin-2-yl)propyl]-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxamide
1-benzyl-N3-cyclopropyl-N5-[1-(4-fluorophenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-ethyl-3-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
6-cyclopentyl-N,1-dimethyl-N-[(3-methylpyridin-4-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-[(1r,4r)-4-methylcyclohexanecarbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(pyridin-2-ylmethyl)piperidin-2-one
4-({4-[(4-chlorophenyl)methyl]piperazin-1-yl}methyl)-2-(propan-2-yl)pyrimidine
(2S,4R)-1-[(5-cyclopentylthiophen-2-yl)methyl]-N-ethyl-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl](methyl)[(6-methylpyridin-2-yl)methyl]amine
5-(pyridin-3-yl)-5-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
6-[4-(piperidin-1-yl)piperidin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(3R,4S)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-N,N-dimethyl-4-propylpyrrolidin-3-amine
1'-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]
4-[3-(2-ethylphenyl)phenyl]-4H-1,2,4-triazole
(1R,5R)-N,N-dimethyl-6-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]benzamide
4-(5-{imidazo[1,2-a]pyridine-2-carbonyl}-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)morpholine
1-[(4aR,8aR)-1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-(2-methoxyphenyl)ethan-1-one
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[(2-chloro-6-fluorophenyl)methyl]-1,4-oxazepan-5-one
3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-{3-[(diethylamino)methyl]phenyl}-3-methylurea
[(3S,5R)-1-(2,5-dimethylfuran-3-carbonyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
1-cyano-N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]cyclopropane-1-carboxamide
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-5-[(dimethylamino)methyl]furan-2-carboxamide
4-ethyl-1-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
[2-(2-methoxypyridin-3-yl)-8-methylquinolin-3-yl]methanol
3-(4-methylphenyl)-3-{[1-(pyrimidin-2-yl)piperidin-4-yl]amino}propan-1-ol
(1H-imidazol-4-ylmethyl)(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(morpholin-3-yl)acetamide
3-(3-acetylphenyl)-6-(2,1,3-benzothiadiazol-5-ylmethyl)-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]-4-methylphenol
methyl({[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl})(quinolin-5-ylmethyl)amine
4-[(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)methyl]morpholine
4-cyclobutaneamido-N-[2-(cyclohex-1-en-1-yl)ethyl]benzamide
6-methyl-3-{[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(3S,9aR)-3-[(4-methoxyphenyl)methyl]-8-(thiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(5-ethylthiophene-3-carbonyl)pyrrolidin-3-yl]methanol
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-2-(2H-1,3-benzodioxol-5-yloxy)acetamide
7-methoxy-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methoxypiperidine
3-(3,5-dimethylphenyl)-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
(2S,4R)-4-{[(3-methylphenyl)methyl]amino}-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide