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6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxylic acid
N-tert-butyl-4-[3-(4H-1,2,4-triazol-4-yl)phenyl]benzene-1-sulfonamide
(3aS,6aS)-2-[2-(2,3-difluorophenyl)acetyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)-1,4-dihydroquinolin-4-one
3-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
N-[1-({[3-(1H-imidazol-1-yl)-1-phenylpropyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
{2H-1,3-benzodioxol-5-yl[1-ethyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}dimethylamine
N-(2-methylpropyl)-1-[(1s,4s)-4-[3-(3-methoxyphenyl)propanamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
ethyl 1-[2-(cyclohex-1-en-1-yl)acetyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
4-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-N-methylpyridin-2-amine
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
3-(1,3-benzothiazol-2-yl)-1-[3-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]propan-1-one
methyl 3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxylate
N-(5-oxo-1-propylpyrrolidin-3-yl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-{2-[1-(4-fluorophenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-(1-methylpiperidin-4-yl)propanamide
1-ethyl-N,4,6-trimethyl-2-oxo-N-(quinolin-5-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-(3-ethyladamantan-1-yl)-3-(1,3,4-thiadiazol-2-yl)urea
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-acetamidoacetamide
2-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-N,N-dimethylaniline
9-(2-cyclopropylquinoline-4-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-[methyl(oxolan-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-[({1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-3-yl}oxy)methyl]pyridine
dimethyl[2-(2-{1-[(3-methylphenyl)methanesulfonyl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
2,3-dimethyl-6-[2-(pyridin-3-yl)piperidine-1-carbonyl]quinoxaline
4-ethyl-1-[2-(naphthalen-1-yl)ethyl]-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-2,8-dimethylquinoline-4-carboxamide
N-[1-(pyridin-4-yl)propyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,3-oxazole-4-carboxamide
[benzyl(methyl)sulfamoyl][1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
3-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-N,N-dimethylpropane-1-sulfonamide
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-(quinoxalin-2-ylmethyl)propanamide
3-[5-({7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)thiophen-3-yl]prop-2-yn-1-ol
2-methyl-N-[(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]butanamide
1-benzyl-8-[(4-methoxyphenyl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{1-[2-(3-fluoro-4-hydroxyphenyl)acetyl]piperidin-3-yl}benzoic acid
4-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
3-(2-fluorophenyl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
methyl 6-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidine-1-carbonyl}pyridine-3-carboxylate
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2,4-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperazine
8-(2-amino-6-methylpyrimidin-4-yl)-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{4-[5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}pyrazine
1-[3-(prop-2-en-1-yloxy)benzoyl]-4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
2-{[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}-3-(thiophen-3-yl)propan-1-ol
[(3-methyl-1H-pyrazol-5-yl)methyl][(2-methylphenyl)methyl](prop-2-en-1-yl)amine
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
2-(2-ethylpyrimidin-5-yl)-7-methyl-4-(2-methylpyrrolidine-1-carbonyl)quinoline