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3-[1-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-hydroxy-2-methylpropyl)acetamide
4-({4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
2,4,6-trimethyl-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)benzamide
7-methyl-3-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-[2-(2-chlorophenoxy)ethyl]-N-ethyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
5-fluoro-2-[3-(piperidin-1-ylmethyl)piperidin-1-yl]pyridine
N-(3-chloro-4-fluorophenyl)-3-{1-[2-(1H-imidazol-2-yl)ethyl]piperidin-4-yl}propanamide
4-{5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]furan-2-yl}-2-methylbut-3-yn-2-ol
1-{1-[1-(1-methylcyclopropyl)propan-2-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
4-(piperidin-1-ylmethyl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}benzamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-3-(4-phenyl-1,2,3-thiadiazol-5-yl)urea
6-methyl-1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-[4-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)phenyl]-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
6-(2-chlorophenyl)-2-(3-hydroxyazetidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
[(2-methoxyphenyl)methyl]({[2-(propan-2-yl)pyrimidin-4-yl]methyl})(pyridin-3-ylmethyl)amine
1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-4-(4H-1,2,4-triazol-3-yl)piperidine
1-(4-ethylpiperazin-1-yl)-3-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}propan-1-one
1-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-(2-phenylethyl)-1H-1,2,3-triazole
{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-(1-cycloheptylpiperidin-3-yl)-2-(diethylamino)acetamide
4-(3-ethyl-4-methylpiperazine-1-carbonyl)-7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
8-[(4Z)-hept-4-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
3-[(5-ethylfuran-2-yl)methyl]-3,9-diazaspiro[5.5]undecane
2-methyl-6-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
2-[2-(dimethylamino)ethyl]-8-[2-methyl-2-(1H-pyrrol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-{[(2S,5R)-5-(pyrrolidin-1-ylmethyl)oxolan-2-yl]methyl}quinoline
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amine
2-(4-fluorophenoxymethyl)-N-[1-(pyridin-4-yl)propyl]-1,3-oxazole-4-carboxamide
5-ethyl-4-[3-(methoxymethyl)piperidin-1-yl]-6-methylpyrimidin-2-amine
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-propylacetamide
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-2-(3-methyl-1,2-oxazol-5-yl)acetamide
5-(3-methoxyphenoxymethyl)-N-(1-propylcyclopropyl)-1,2-oxazole-3-carboxamide
(1R,6S)-3-{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-9-methyl-3,9-diazabicyclo[4.2.1]nonane
(3aS,6aS)-2-(2-hydroxyethyl)-5-{[4-(propan-2-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[1-(methoxymethyl)cyclopentyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)cyclohexanecarboxamide
N-benzyl-1-(2-hydroxyethyl)-5-{[5-(methoxymethyl)furan-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-[5-(methoxymethyl)furan-2-carbonyl]-7-methyl-4-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
1-ethyl-4-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
6-[({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)amino]-N-ethylpyridine-3-carboxamide
{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(trifluoromethyl)phenyl]methyl}amine
ethyl 4-{[4-(3-phenyl-1,2-oxazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazine-1-carboxylate
2-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}-4-hydroxyquinoline-6-carboxamide
2-{2-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}-2-azaspiro[4.5]decan-3-one
2-(4-methyl-2-oxo-1,2-dihydroquinolin-1-yl)-N-(3-phenylprop-2-yn-1-yl)-N-propylacetamide
3-(3-hydroxy-1,2-oxazol-5-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}propanamide