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N'-(3,5-dimethylphenyl)-N-methyl-N-(2-methylprop-2-en-1-yl)propanediamide
N-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyloxolan-3-amine
1-(4-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)ethan-1-one
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-3-phenyl-1H-pyrazole-5-carboxamide
4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-1,2,3,6-tetrahydropyridine
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-(2-cyclohexylethyl)-N-[(6-methylpyridin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-{1-[2-(2H-1,3-benzodioxol-5-yloxy)acetyl]piperidin-3-yl}benzoic acid
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
(3S,4R)-1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}benzenesulfonamide
9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
(2-methoxyethyl)({[(2R,5S)-5-[(5-methoxypyridin-3-yl)methyl]oxolan-2-yl]methyl})methylamine
2-[(3,4-difluorophenyl)methyl]-8-(1,3-thiazol-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
2-(2-methoxyphenyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
methyl 1-[(3R,5S)-1-[(4-ethoxyphenyl)methyl]-5-(4-phenylpiperazine-1-carbonyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-2-methylphenol
6-{[3-(diethylcarbamoyl)piperidin-1-yl]methyl}-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
7-[(2-methoxypyrimidin-5-yl)methyl]-N,2-dimethyl-N-(prop-2-en-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}cyclopentanamine
2-(dimethylamino)-2-(3-methylphenyl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(dimethyl-1,2-oxazol-4-yl)methyl]propanamide
5-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
(3R,4R)-1-cyclobutanecarbonyl-4-({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)pyrrolidin-3-ol
N4-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N1,N1-dimethylpiperidine-1,4-dicarboxamide
3-{[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]sulfonyl}benzoic acid
1-[7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
4-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-1-(2-methylphenyl)piperazin-2-one
3-methoxy-1-{4-[4-(3-methoxypiperidine-1-carbonyl)phenoxy]piperidin-1-yl}propan-1-one
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
(1R,5R)-6-(2-methoxyethyl)-3-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
1-(2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholin-4-yl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
2-hydroxy-1-[4-(3-methylphenoxy)piperidin-1-yl]-4-(methylsulfanyl)butan-1-one
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]pyrimidin-4-amine
4-(2,4-dioxoimidazolidin-1-yl)-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}benzamide
2-(3,4-dichlorophenyl)-4-(3-propyl-1H-pyrazole-4-carbonyl)morpholine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]propan-1-one
N-[2-(ethanesulfonyl)ethyl]-3-(4-methylphenyl)-1H-pyrazole-5-carboxamide
2-fluoro-N-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-sulfamoylbenzamide
N-[1-(7-{[4-(dimethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-3-methylbutyl]-5-(methoxymethyl)furan-2-carboxamide
1-[7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(4-methylphenyl)propan-1-one
N,N-dimethyl-4-[4-({[2-(trifluoromethyl)phenyl]methyl}amino)piperidin-1-yl]benzamide
7-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-1,2-dihydroisoquinolin-1-one
6-[9-oxo-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-2-carbonitrile