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N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-1,3-thiazole-5-carboxamide
7-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
3-[(dimethylamino)methyl]-N-[1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]benzamide
2-(2-chlorophenoxy)-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
methyl({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})[(5-phenyl-1H-pyrazol-4-yl)methyl]amine
N-ethyl-4-[4-(piperidin-3-yl)benzamido]piperidine-1-carboxamide
N-(2-{[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}quinolin-6-yl)acetamide
3-oxo-2-(oxolan-2-ylmethyl)-N-(2-phenylethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-{3-cyclopentyl-5-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazol-4-yl]-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
2-{[3-({3-[(pyridin-3-yl)amino]propyl}carbamoyl)phenyl]amino}acetic acid
[(2S,6S)-11-methoxy-4-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
(3aS,7aR)-5-methyl-2-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-[(3E)-hex-3-enoyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
1-(oxolane-2-carbonyl)-N-(pentan-3-yl)-N-(2-phenylethyl)piperidine-4-carboxamide
1-(1H-indazol-6-yl)-5-methyl-4-(5-methylpyrazine-2-carbonyl)piperazin-2-one
N-(1,4-dioxan-2-ylmethyl)-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
1-(2-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)piperidin-2-one
4-[(2S)-2-amino-3-phenylpropanamido]-N-(2,6-dimethylphenyl)benzamide
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[(3-methylpyridin-2-yl)methyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-methyl-1-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(1H-1,2,4-triazol-3-yl)urea
2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}quinoxaline
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
8-[4-(benzyloxy)butyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]pent-4-enamide
4-{cyclopropyl[(3-hydroxyphenyl)methyl]carbamoyl}benzoic acid
1-[1-(propan-2-yl)pyrrolidine-3-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(1-phenylcyclopentanecarbonyl)pyrrolidin-3-yl]methanol
1-(pyridin-3-ylmethyl)-4-[5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,4-diazepane
8-methoxy-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(1S,5R)-6-(4-chloro-2-fluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-2-(propan-2-yl)pyrimidine-5-carboxamide
3-(3-methyl-1,2,4-oxadiazol-5-yl)-1-(oxan-4-yl)piperidine
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-[(3-hydroxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]acetamide
ethyl 2-({[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)amino)acetate
N-[2-({[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]acetamide
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(piperidin-1-yl)acetamide
N-[3-(3-ethylphenoxy)propyl]-N-methyl-1H-imidazole-5-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1H-imidazole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S)-2-[(4-methyl-1,3-thiazol-5-yl)formamido]-3-phenylpropanamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
4-(2-methoxyethoxy)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
N-({3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl}methyl)acetamide
N1-(propan-2-yl)-N2-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-1,2-dicarboxamide
[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
1-[4-({4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
4,4,4-trifluoro-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
(1R,3S)-7-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-ethoxy-7-azaspiro[3.5]nonan-1-ol
1-{2-[4-(3-cyanophenyl)piperidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide