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3-(1-methyl-1H-imidazole-2-carbonyl)-1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperidine
3-(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)phenol
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]propan-1-one
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
(2S)-N-{[5-chloro-7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-oxopyrrolidine-2-carboxamide
N,1-dimethyl-6-(pyridin-3-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyridin-1-ium-1-olate
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
[1-(2-chlorophenyl)-2-[2-(furan-3-yl)-1H-imidazol-1-yl]ethyl]dimethylamine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-{[7-(2H-1,3-benzodioxole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-sulfonamide
5-ethyl-2,3-dimethyl-N-[1-(pyridin-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
(2S,4S)-4-{4-[2-(furan-2-ylformamido)propan-2-yl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
5-[({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
2-{2-[2-(benzylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}acetamide
4-[4-(4-ethylphenyl)-1H-imidazol-2-yl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
N-[2-(1H-imidazol-4-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-methyl-N-[(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]piperidine-3-carboxamide
2-{[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
[4-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)piperidin-4-yl]methanol
2-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-2,3-dihydro-1H-isoindole
(1R,5R)-6-(8-fluoro-4-oxo-1,4-dihydroquinoline-3-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[(3-methyl-1H-indol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
1-[(2-chloro-6-fluorophenyl)methyl]-5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-3-methyl-1H-1,2,4-triazole
5-{[1-(3-methylbut-2-enoyl)pyrrolidin-3-yl]methyl}-1,2-dihydropyridin-2-one
3-(1H-1,3-benzodiazol-1-yl)-1-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]propan-1-one
2-amino-4-methyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1,3-benzothiazole-6-carboxamide
3-(5-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
3-(pyrrolidine-1-carbonyl)-1-[1-(thiophene-3-carbonyl)piperidin-4-yl]piperidine
4-(2,2-dimethylpropyl)-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]piperazin-2-one
2-(hydroxymethyl)-N-[(1R,2S)-2-phenylcyclopropyl]-1H-1,3-benzodiazole-5-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-methylthiophene-2-carboxamide
1-{1-[2-(2-chlorophenyl)acetyl]piperidin-3-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
3-methyl-4-[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]oxolan-2-one
[3-(2-{[(propan-2-yl)amino]methyl}phenyl)phenyl]methanol
4-{[2-(6-ethoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]methyl}-1,3-thiazol-2-amine
5-[3-(diethylcarbamoyl)piperidine-1-carbonyl]-1H-imidazole-4-carboxylic acid
3-(1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
4-hydroxy-N-(oxan-4-yl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2-{2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
N-(1-cycloheptylpiperidin-3-yl)-2,3,4-trimethoxybenzamide
N-({1-[(6-ethoxypyridin-3-yl)methyl]piperidin-4-yl}methyl)-2,2-difluoroacetamide
N-methyl-3-(2-methylphenyl)-3-phenyl-N-(pyridin-2-ylmethyl)propanamide
[(5-{2-[(3-fluorophenyl)methyl]morpholine-4-carbonyl}furan-2-yl)methyl]dimethylamine
3,5-difluoro-2-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridine
N-phenyl-3-({[2-(1H-pyrazol-1-yl)ethyl]carbamoyl}methyl)morpholine-4-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[1-(4-fluorophenyl)ethyl]benzamide