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N-[(3-fluorophenyl)methyl]-5-methyl-6-(piperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
3-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenol
N-cyclopentyl-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
4-{5-methyl-4-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl}-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
N-[(3R,4S)-4-cyclopropyl-1-(3-methylthiophene-2-carbonyl)pyrrolidin-3-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-3-(morpholin-4-yl)propanamide
N-(2-methanesulfonylethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-fluoro-4-methyl-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)benzamide
[1-({[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl](methyl)amino}methyl)cyclopropyl]methanol
N-methyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-(pyrimidin-4-ylmethyl)acetamide
N,6-dimethyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(3S,9aR)-3-[(4-methoxyphenyl)methyl]-8-(2,4,5-trifluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
[(4-methanesulfonylphenyl)methyl][(3-methoxyphenyl)methyl](prop-2-en-1-yl)amine
2-amino-1-{4-[(2-aminopyridin-3-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}-2-methylpropan-1-one
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
1-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]sulfonyl}azepane
methyl 3-(oxolane-2-amido)-1-(2-phenylethyl)-5-[(thiolan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1R,2S,9R)-11-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
2-methyl-5-{3-[({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]pyrrolidin-1-yl}-2,3-dihydropyridazin-3-one
4-ethyl-3-[(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-({2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)benzonitrile
N-(1-methyl-1H-indazol-3-yl)-2-[3-(5-methylthiophen-2-yl)-1H-pyrazol-1-yl]acetamide
3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-N-(2-fluorophenyl)propanamide
N-[(3,4-difluorophenyl)methyl]-3-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}propanamide
N-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-[(3-fluorophenyl)methyl]-N-methyl-N-[(3-methylpyridin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
2-[2,4-dioxo-1,8-bis(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
2-(2-methoxy-5-methylphenyl)-2-[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]acetic acid
3-(3-hydroxyquinoxalin-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}propanamide
4-(4-phenyl-1H-pyrazol-5-yl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
2-(4-fluoro-3-methylphenyl)-2-{methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}acetic acid
2-methyl-5-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}phenol
4-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-methyl-6-(propan-2-yl)pyrimidine
3-[2-({[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-1,3-oxazolidin-2-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
7-(5-methylthiophen-2-yl)-4-(oxolane-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(1H-imidazol-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-N2-(3-methylphenyl)-1,3,5-triazine-2,4-diamine
4-{[2-(4-chlorophenyl)-7-methoxyquinolin-3-yl]methyl}-3-methylpiperazin-2-one
(3S,4R)-4-phenyl-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}pyrrolidine-3-carboxylic acid
2-[4-(6-chloroquinolin-2-yl)-1-(1-methylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
4-(4-methyl-1H-pyrazol-1-yl)-1-(4-methylpyrimidin-2-yl)piperidine-4-carboxylic acid
1-methyl-4-({5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)piperazine
N-[3-(1,4-oxazepane-4-carbonyl)phenyl]pentanamide
N-(3-hydroxy-2,2-dimethylpropyl)-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
5-{[benzyl(methyl)amino]methyl}-N-(1-methylpiperidin-4-yl)-1,2-oxazole-3-carboxamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
2-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-1H-1,3-benzodiazole
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-(2-methylphenyl)pyrrolidin-3-ol