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2-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
8-(2-hydroxyethyl)-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4S)-1-[(2,5-dimethylphenyl)methyl]-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-2-(1H-imidazol-4-yl)-N-methylacetamide
N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrrole-2-carboxamide
N-cyclopropyl-5-[2-(2H-indazol-2-yl)acetyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
5-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}pyrazin-2-ol
4-[(4-methoxyphenyl)methyl]-3-(pyridin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2R,3R)-2-(prop-2-en-1-yloxy)-1'-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]cyclopropanecarboxamide
4-{4-[3-(2-methoxyethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
7-(2-chloro-6-fluoro-3-methylbenzoyl)-3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine
5-(azepane-1-carbonyl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-1-benzoxepine-4-carboxamide
3-chloro-N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}pyridine-4-carboxamide
1-[1-(6-aminopyridine-3-carbonyl)piperidin-3-yl]pyrrolidin-2-one
9-(1-methyl-1H-pyrazole-4-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-phenyl-5-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-1,2,4-oxadiazole
2-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
2-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-N-(4-methylphenyl)-2-oxoacetamide
1-[2-chloro-5-(trifluoromethyl)benzoyl]-4-(1-ethyl-1H-imidazol-2-yl)piperidine
N-[(3R,4S)-1-(3-hydroxypropyl)-4-propylpyrrolidin-3-yl]-1H-1,2,3-triazole-5-carboxamide
2-(azetidine-1-carbonyl)-6-chloro-1-methyl-1H-indole
(1R,5S,6S)-6-{[4-(2-phenylethyl)piperidin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
5-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]-2-(methylsulfanyl)pyrimidine
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidine-3-carboxylic acid
1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-8-{[2-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(piperidin-1-yl)piperidine
1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(4-fluorophenyl)piperazine
1-cyclopropyl-4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-5-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(3R,4R)-3-cyclobutyl-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-methylpyrrolidin-3-ol
(1S,6R)-9-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonane
2-[2-(1H-pyrazol-1-yl)ethyl]-1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine
2,3-dimethyl-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]-1H-indole-7-carboxamide
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
(2S,4R)-4-amino-1-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-N-methylpyrrolidine-2-carboxamide
(1R,5R)-6-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(2,3-dihydro-1H-isoindole-2-carbonyl)-3,4,7-trimethyl-1H-indole
2-({[(3R,4R)-1-[4-(dimethylamino)benzoyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
methyl 4-(5-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
methyl 5-(cyclopentylamino)-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1R,5R)-3-benzoyl-6-[(2-fluoro-5-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
methyl 3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-5-[(1,3-thiazol-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
methyl({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)[1-(pyrimidin-4-yl)ethyl]amine
(2S,4R)-N-[2-(4-fluorophenyl)ethyl]-1-[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
4-{2-methyl-6-[1-(2-methylpyrimidine-5-carbonyl)piperidin-3-yl]pyrimidin-4-yl}morpholine
[(3-ethoxy-4-methoxyphenyl)methyl](methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
1-[(2-chlorophenyl)methyl]-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide