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1-{[(2R,5S)-5-(2H-1,3-benzodioxol-5-ylmethyl)oxolan-2-yl]methyl}-4-methylpiperazine
N,3,5-trimethyl-N-[1-(pyrimidin-4-yl)ethyl]adamantane-1-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]pyrrolidin-3-yl]-3-methoxypropanamide
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(3,3,3-trifluoropropyl)amine
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}pyrrolidin-3-yl]methanol
2-(4-fluorophenoxy)-1-(3-propylmorpholin-4-yl)ethan-1-one
N-({5-[3-(dimethylamino)pyrazin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
{1-[2-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]piperidin-2-yl}methanol
4-[1-(4-chloro-1H-pyrrole-2-carbonyl)piperidin-4-yl]thiomorpholine
(3S,4R)-1-(4-hydroxybenzoyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(oxan-2-ylmethoxy)acetamide
6-methyl-2-[2-({methyl[(2E)-3-phenylprop-2-en-1-yl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]methylamine
[(3-chloro-4,5-dimethoxyphenyl)methyl]({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-(1-{4-[(2S)-4-ethyl-2-methyl-3-oxopiperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)furan-3-carboxamide
methyl 2-({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}sulfamoyl)benzoate
3,5-dimethyl-2-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}-1H-indole
8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 4-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}piperazine-1-carboxylate
1-(cyclopropylmethyl)-4-(6-methylpyridine-3-carbonyl)-2-(propan-2-yl)-1,4-diazepane
N-(cyclohexylmethyl)-4-(3-hydroxypyrrolidine-1-carbonyl)benzene-1-sulfonamide
2-(benzyloxy)-N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
4-(piperidin-1-yl)-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
1-[(3-fluorophenyl)methyl]-6-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}piperidine-3-carboxamide
N-(2-{1-[2-(2-chloro-5-methylphenoxy)-2-methylpropanoyl]piperidin-4-yl}ethyl)acetamide
methyl 6-[(1-hydroxybutan-2-yl)(thiophen-3-ylmethyl)carbamoyl]pyridine-3-carboxylate
3-(dimethyl-1,2-oxazol-4-yl)-1-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}propan-1-one
(4R)-4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-3-methyl-1,3-thiazolidine
methyl 4-(5-chloro-2-{[(4-methyl-1,2,3-thiadiazol-5-yl)formamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(phenylsulfanyl)acetamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(4-hydroxyphenyl)ethyl]acetamide
(2S)-2-{[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]amino}-3-(4-hydroxyphenyl)propanamide
3-[(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)oxy]pyridine
1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3-propoxypiperidine
N-(furan-3-ylmethyl)-N-methyl-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-(oxolan-3-yl)-1H-pyrazole-3-carboxamide
(3R,4R)-4-ethyl-1-[5-(ethylsulfanyl)thiophene-2-carbonyl]piperidine-3,4-diol
1-(4-{[2-(1H-imidazol-4-yl)ethyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-(3-{[({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(2-methylpropyl)amino]methyl}phenoxy)ethan-1-ol
1-{4-[(3-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}-4-methoxyphenyl)methyl]piperazin-1-yl}ethan-1-one
N-(3-hydroxypropyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
2-(1-methyl-4-{[4-(5-methylfuran-2-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
1-[cyclohexyl(methyl)amino]-3-{3-[(4-fluoropiperidin-1-yl)methyl]phenoxy}propan-2-ol
(3aR,6aR)-2-acetyl-5-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)benzamide
2-methyl-N-{[3-methyl-7-(4-methylpentanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}furan-3-carboxamide
2-[(5-ethylfuran-2-yl)methyl]-9-oxa-2-azaspiro[5.5]undecane
7-[(3-methoxyphenyl)methyl]-2-(5-methyl-1H-indazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
2-(4-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}piperidin-1-yl)ethan-1-ol