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N,N-dimethyl-5-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}pyridin-2-amine
1-(4-fluorophenyl)-6,6-dimethyl-N-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-[(3-methoxyphenyl)methyl]-3-methyl-5-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
[(3R,4R)-1-[2-amino-6-(dimethylamino)pyrimidin-4-yl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-4-hydroxy-2-(3-methylphenyl)pyrimidine-5-carboxamide
4-[(1-{[1-(1-methylcyclohexanecarbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
methyl({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl})[2-(1H-pyrazol-4-yl)ethyl]amine
4-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-phenylpiperazin-2-one
N-(cyclohexylmethyl)-5-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
{1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-2-phenylethyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
(2-ethoxy-5-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}phenyl)methanol
5-(2-fluorophenoxymethyl)-N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-1H-pyrazole-3-carboxamide
6-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}pyridine-2-carbonitrile
N-[1-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
4-fluoro-N-(2-{[2-(1H-imidazol-2-yl)phenyl]formamido}ethyl)benzamide
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
5-cyclopropanecarbonyl-1'-[(5-methylthiophen-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(3-fluoro-4-hydroxyphenyl)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(4-methylpent-3-en-1-yl)piperidine
2-(4-chlorophenyl)-4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)morpholine
2-({4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazin-1-yl}methyl)quinolin-4-ol
N-{[5,8-dimethoxy-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]furan-2-carboxamide
N,N-dimethyl-2-[1-(1H-1,2,3,4-tetrazol-5-yl)-1H-pyrazol-4-yl]aniline
N-[3-({[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]carbamoyl}methoxy)phenyl]propanamide
2-(3-fluorophenyl)-2-hydroxy-N-methyl-N-{2-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
N-[3-(4-cyanopyridin-2-yl)phenyl]acetamide
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2,5-dimethylbenzamide
1-(2-{[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]amino}pyrimidin-4-yl)piperidin-3-ol
N-[(2-ethoxyphenyl)methyl]-3-fluoro-8-methyl-N-(prop-2-en-1-yl)imidazo[1,2-a]pyridine-2-carboxamide
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-{2-[3-methyl-1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(2-methoxyethyl)-5-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
N-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-ethyl-N-[(2-methoxyphenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3,4-dimethoxy-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
2-methyl-N-(2,4,5-trifluorophenyl)-2,7-diazaspiro[4.5]decane-7-carboxamide
1-[(2-chloro-6-fluorophenyl)methyl]-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N,6-dimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
2,3,5,6-tetramethyl-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]benzamide
N-[(3R,4S)-4-cyclopropyl-1-[(2-methylphenyl)methyl]pyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
N-{1-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]ethyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
[2-(1H-1,3-benzodiazol-2-yl)ethyl](methyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
1-[1-(thiophen-3-yl)propan-2-yl]-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
3-fluoro-N-[2-(1H-imidazol-4-yl)ethyl]-5-methylimidazo[1,2-a]pyridine-2-carboxamide
3-[(1R,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-N-(isoquinolin-5-ylmethyl)-N-methylpyridin-2-amine
N-{[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-4-yl)piperazine
2-(2,6-dimethylquinoline-4-carbonyl)-1,2-oxazolidin-4-ol
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]acetamide
N-[3-({[2-(1-benzylpyrrolidin-3-yl)ethyl]carbamoyl}amino)phenyl]acetamide