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5-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(furan-2-carbonyl)piperidin-3-ol
N-[1-(2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetyl)piperidin-4-yl]methanesulfonamide
8-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 2-{2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-methylacetamido}acetate
1-(2-ethoxypyridine-3-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-2-methyl-1,4-diazepan-5-one
1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-(3,4-dimethylphenoxy)ethan-1-one
N-(8-chloroquinolin-5-yl)-3-[(methylsulfanyl)methyl]piperidine-1-carboxamide
5-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
1,6-dimethyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-[6-methyl-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carbonyl]-1-oxa-8-azaspiro[4.5]decane
2-cyclopropyl-N-[4-(furan-2-yl)butan-2-yl]-4-hydroxypyrimidine-5-carboxamide
N-[(3S,4R)-1-(4-phenylbenzoyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-chloro-6-fluoro-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}benzamide
5-benzyl-5-(piperidin-4-yl)-3-(pyrazin-2-ylmethyl)imidazolidine-2,4-dione
1-[3-(4-tert-butylbenzoyl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-3-hydroxy-2-methylbenzamide
1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyrrolidin-1-yl)piperidine
methyl 5-({[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}amino)-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(1H-indol-5-ylmethyl)-4-(1,2-oxazole-3-carbonyl)-1,4-diazepan-6-ol
1-[(2S,4S)-1-{[3-(4-chlorophenoxy)phenyl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carbonyl]azepane
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
8-(3,5-dichloro-4-methylbenzoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[4-(butan-2-yl)phenyl]-3-[3-(1H-imidazol-2-yl)propyl]urea
3-{[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)amino}propane-1,2-diol
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(1-methyl-1H-pyrazol-4-yl)-N-(propan-2-yl)quinoline-4-carboxamide
2-[ethyl(oxan-4-yl)amino]-N-[(2-methoxyphenyl)methyl]acetamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1-ethylpyrrolidine-3-carboxamide
(1S,4S)-2-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-azabicyclo[2.2.1]heptane
3,4,7-trimethyl-2-[(2S)-2-(piperidine-1-carbonyl)pyrrolidine-1-carbonyl]-1H-indole
2-(3-phenylpropyl)-4-(1,3-thiazol-2-ylmethyl)morpholine
2-{1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]piperidin-4-yl}ethan-1-ol
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(2-phenylpropan-2-yl)amino]methyl}piperidin-2-one
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-methoxypropan-1-one
3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}(methyl)amino)-N-methylbutanamide
1-tert-butyl-N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-1H-pyrrole-3-carboxamide
3-(1-butyl-1H-imidazol-2-yl)-1-(2-chloro-6-fluoro-3-methylbenzoyl)piperidine
4-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(2-methoxypyridin-3-yl)-N-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
2-[(isoquinolin-5-yloxy)methyl]-N-[2-(6-methylpyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
1-[(2,3-difluorophenyl)methyl]-4-[(3-methoxyphenyl)methyl]-1,4-diazepan-5-one
(2,1,3-benzothiadiazol-5-ylmethyl)({[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl})methylamine
3-hydroxy-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-(cyclohexylmethyl)-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-1,3-thiazole
6-methyl-5-{2-oxo-2-[4-(4H-1,2,4-triazol-3-ylmethyl)piperazin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2,2-dimethyl-N-({1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-yl}methyl)propanamide
5-{[4-(diphenylmethyl)piperazin-1-yl]methyl}-2-ethylpyrimidine