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N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
(1R,5R)-N,N-dimethyl-6-(5-propyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
6-[2-(2-aminoethyl)morpholin-4-yl]-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-amine
1-{4-[(dimethylsulfamoyl)amino]phenyl}-N-[2-(thiophen-2-yl)ethyl]piperidin-4-amine
1-methyl-3-(2-methylpropyl)-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 4-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamido]piperidine-1-carboxylate
3-[4-(propylsulfamoyl)phenyl]-1-[1-(pyridin-3-yl)propan-2-yl]urea
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
(3S)-N,N-dimethyl-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)azepan-3-amine
2-{5-[2-(hydroxymethyl)-1H-1,3-benzodiazol-5-yl]-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylfuran-2-carboxamide
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]acetamide
4-ethyl-1-methyl-3-(1-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-2,8-dimethylquinoline-4-carboxamide
(2S)-2-cyclohexyl-2-{[1-ethyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}acetic acid
N-cyclohexyl-4-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-N-methylpyridine-2-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
4-[(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)methyl]morpholine
[2-({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-1,3-thiazol-4-yl]methanol
2-{3-[(4-fluorophenyl)methoxy]phenyl}-4-(pyrrolidine-1-carbonyl)pyridine
2,6-dimethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}quinoline-3-carboxamide
3,5-dimethyl-2-{[5-(1-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyridin-4-ol
3-chloro-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-4-fluoro-1-benzothiophene-2-carboxamide
2-[4-(dimethyl-1,3-oxazole-5-carbonyl)-6-hydroxy-1,4-diazepan-1-yl]acetic acid
2-{4-[(cyclopent-3-en-1-yl)amino]-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}acetic acid
2-methyl-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-1-benzofuran-7-carboxamide
4-[5-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
[(2S,4R)-4-(dimethylamino)-1-[(2-methoxynaphthalen-1-yl)methyl]pyrrolidin-2-yl]methanol
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
4-(2-ethylpyrimidine-5-carbonyl)-N,N-dimethylpiperazine-1-carboxamide
dimethyl({[(1R,5S,6S)-3-[(5-phenylthiophen-2-yl)methyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(2,4-difluorophenoxy)ethan-1-one
3-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-N-(1,3-thiazol-2-yl)propanamide
N-[(4-methoxyphenyl)methyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
8-(5-{6-azaspiro[2.5]octan-1-yl}-3-methyl-1H-1,2,4-triazol-1-yl)quinoline
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-4-(pyrrolidin-1-yl)butan-1-one
(1R,5R)-3-(5-chloro-3-methyl-1H-indole-2-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 4-[({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)carbamoyl]butanoate
N-({1-[(2-methoxynaphthalen-1-yl)methyl]pyrrolidin-3-yl}methyl)methanesulfonamide
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl 1-[(3S,5S)-1-(adamantan-2-yl)-5-{[(4-methoxyphenyl)methyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
ethyl 1-(2-methoxybenzoyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-(2,3-dihydro-1H-inden-2-yl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
(2R)-2-acetamido-N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}butanamide
3-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2,5-dimethylpyrazine
5-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}-3-phenyl-1,2,4-oxadiazole
ethyl 2-{1-[6-oxo-1-(2-phenylethyl)piperidine-3-amido]cyclohexyl}acetate
3-[(1-methylazepan-2-yl)formamido]-N-phenylpropanamide
N-(1-{7-[(3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide