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(2S,4S)-1-benzyl-4-{[(2-chlorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-ethyl-3-(naphthalen-2-yl)-1-(oxan-4-ylmethyl)urea
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
methyl (2R,4S)-1-[(3-chloro-4-ethoxyphenyl)methyl]-4-hydroxypiperidine-2-carboxylate
ethyl 2-(1-{3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanoyl}piperidin-2-yl)acetate
3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
2-(adamantan-1-yl)-5-{2,8-diazaspiro[4.5]decane-2-carbonyl}pyrimidin-4-ol
methyl 5-[4-(2-methylpropyl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[(3,4-difluorophenyl)methyl]-3-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-3-yl}propanamide
(1S,5S)-N-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
methyl 4-({2-methyl-2,8-diazaspiro[4.5]decane-8-carbonyl}amino)benzoate
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]acetamide
(1R,5R)-6-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-cyclopropyl-2-({1-[(4-hydroxyquinolin-2-yl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
3-methyl-2-oxo-N-phenyl-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
1-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-3-methylbut-2-en-1-one
N-[(2R,3R)-2-methoxy-1'-[2-(1H-1,2,4-triazol-1-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
4-chloro-N-(2-methanesulfonamidoethyl)-2-propanamidobenzamide
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(furan-2-carbonyl)piperidine
{[(1R,5S,6S)-3-(1H-indol-4-ylmethyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
3-{[(4-fluorophenyl)methyl](3-hydroxypropyl)carbamoyl}benzoic acid
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(trifluoromethyl)phenyl]urea
9-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 3-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)butanoate
N-(2-methoxyethyl)-1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
1-cyclohexyl-N3,N5-dimethyl-4-oxo-N3-[1-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-2-methyl-4-phenylpiperazine
ethyl(methyl)[({1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}methyl)sulfamoyl]amine
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-ethyl-6-oxopiperidine-3-carboxamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-(1H-pyrazol-1-yl)butanamide
3-(3-methoxypropyl)-1-(2-methyl-1-benzofuran-5-carbonyl)piperidine
2-methyl-4-[2-(2-phenylethyl)pyrrolidin-1-yl]-6-(piperidin-4-yl)pyrimidine
ethyl 4-{4-[4-({imidazo[1,2-a]pyridin-3-ylmethyl}amino)piperidin-1-yl]benzoyl}piperazine-1-carboxylate
methyl 5-[(2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}acetamido)methyl]furan-2-carboxylate
2-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyridine-3-carboxamide
1-(2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)piperidin-4-ol
1-{2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[1-(1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
1-methoxy-8-[2-(4-methylphenyl)quinoline-4-carbonyl]-1,8-diazaspiro[4.5]decan-2-one
4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(morpholin-4-yl)pyrimidin-2-amine
1-{4-[(2-chlorophenyl)methyl]-5-oxo-1,4-diazepan-1-yl}-4-(4-fluorophenyl)butane-1,4-dione
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methyloxane-2-carboxamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-[(2-phenylphenyl)methyl]piperidin-3-yl]methanol
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-ol
2-(3-{4-[(4-methylphenyl)methyl]-3-oxopiperazine-1-carbonyl}piperidin-1-yl)acetamide
4-[5-(2-aminoethyl)-2-methoxyphenyl]benzamide
methyl 3-(7-chloro-2-{[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetamido]methyl}-2,3-dihydro-1-benzofuran-5-yl)benzoate
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(2,3-dihydro-1H-inden-1-yl)acetamide
1-butyl-4-(5-ethyl-1,3,4-oxadiazol-2-yl)piperazin-2-one