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2-{1-[1-(2,4,5-trifluorobenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
3-[3-({2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)-1H-indol-1-yl]propanamide
7-(cyclopropylmethyl)-2-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(4-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
1-[6-hydroxy-4-(pyridin-4-yl)-1,4-diazepan-1-yl]-2-(thiophen-2-yl)ethan-1-one
N-(1,4-dimethyl-1H-pyrazol-5-yl)-3-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)benzamide
N,6-di-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(2-hydroxyethyl)-3-{[(4-methylphenyl)methyl]amino}-N-(1,3-thiazol-2-ylmethyl)benzamide
dimethyl[1-(pyridin-2-yl)-2-[2-(pyridin-2-yl)-1H-imidazol-1-yl]ethyl]amine
2-(1-{1-[(2,3-dimethylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
4-[(2-fluorophenyl)methyl]-1-(1,3-thiazol-4-ylmethyl)piperidine
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-ol
(1S,5R)-6-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
1-methyl-N-[3-(propan-2-yloxy)propyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(4-methoxy-4-phenylpiperidin-1-yl)-3-(1-methylpiperidin-2-yl)propan-1-one
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methylbutan-1-one
4-{[4-(3-methyl-1-phenyl-1H-1,2,4-triazol-5-yl)furan-2-yl]methyl}morpholine
N-[(3,4-difluorophenyl)methyl]-2-(1H-pyrazol-1-yl)butanamide
N-methyl-3-{1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
5-[3-(3-methylphenyl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
(3S)-4-[2-chloro-5-(piperidin-1-yl)benzoyl]-3-ethylmorpholine
5-(2,3-dihydro-1-benzofuran-2-carbonyl)-3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-({6-methylthieno[2,3-d]pyrimidin-4-yl}sulfanyl)ethan-1-one
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)cyclopropanecarboxamide
1-{3-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(diphenylmethyl)-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
6-ethyl-N-[2-(morpholin-4-yl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
(3S,4R)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
2-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-4-oxo-1,4-dihydroquinoline-8-carboxamide
3-({[(1-benzyl-1H-pyrazol-4-yl)methyl]amino}methyl)-3-hydroxy-1-methylpiperidin-2-one
2-({[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)amino)-1-phenylethan-1-ol
N-[2-(4-fluorophenyl)ethyl]-3-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1,2-oxazole-5-carboxamide
6-methyl-5-[5-(5-methyl-1,2-oxazol-3-yl)-1,2,4-oxadiazol-3-yl]-N-(propan-2-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
2-amino-4-(1,5-dimethyl-1H-pyrazol-4-yl)-6-(4-fluorophenyl)-5-methylpyridine-3-carbonitrile
4-({4-[5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)-N,N-dimethylaniline
1-(2-amino-5-ethylpyrimidin-4-yl)-4-(4-fluorophenyl)piperidin-4-ol
3-(1-ethyl-1H-imidazol-2-yl)-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidine
1-{2-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}pyrrolidin-2-one
[4-(1-phenylcyclohexanecarbonyl)-1,4-oxazepan-6-yl]methanol
1-(morpholin-4-yl)-3-{3-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxy}propan-2-ol
N-[(5-chlorothiophen-2-yl)methyl]-2-(dimethylamino)-2,3-dihydro-1H-indene-2-carboxamide
2-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)quinoline
N-(2-fluoro-5-methylphenyl)-2-[2-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carboxamide
4-cyano-N-[2-(dimethylamino)-1-phenylethyl]-N,1-dimethyl-1H-pyrrole-2-carboxamide
ethyl 1-(2-methoxyethyl)-5-[2-(phenylsulfanyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
methyl 4-(4-{4-[(pyridin-2-ylmethyl)carbamoyl]phenoxy}piperidin-1-yl)pentanoate
1-[(5-ethylfuran-2-yl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
N-{2-[7-(furan-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-methylpropanamide
ethyl 4-[(4-methoxyphenyl)methyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidine-4-carboxylate