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1-(2-chlorophenyl)-4-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)pyrrolidin-2-one
2-[2,4-dioxo-1-(2-phenylethyl)-8-(quinolin-7-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{3-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}acetamide
4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-1-(2-methylfuran-3-carbonyl)piperidine
2-(2-chloro-4-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}phenoxy)acetamide
methyl({3-[(4-methylphenyl)sulfanyl]propyl}){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
[1-(2,3-dihydro-1H-inden-2-yl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
9-[(2-methylpyrimidin-5-yl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[3,5-bis(trifluoromethyl)phenyl]-4-hydroxy-N-methyl-N-(prop-2-yn-1-yl)pyrimidine-5-carboxamide
2-amino-6-[4-fluoro-2-(trifluoromethyl)phenyl]-4-(piperidin-4-yl)pyridine-3-carbonitrile
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}quinoline-3-carboxamide
1-(4-{[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]sulfonyl}phenyl)ethan-1-one
8-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-1-[3-(phenylamino)piperidin-1-yl]propan-1-one
1,5-dimethyl-2-phenyl-4-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-2,3-dihydro-1H-pyrazol-3-one
1-(2,3-dimethylquinoxaline-6-carbonyl)-N-(furan-2-ylmethyl)piperidine-4-carboxamide
6-({4-[1-(3-methylpyridin-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-cyclohexyl-2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N-methylacetamide
(1S,3R)-3-{[methyl(phenyl)carbamoyl]amino}-N-[(5-methylpyrazin-2-yl)methyl]cyclopentane-1-carboxamide
N3-cyclooctyl-N5-[3-(dimethylamino)-2,2-dimethylpropyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[4-(1H-indole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-4-(1H-pyrazol-1-yl)butan-2-ol
(3R,9aR)-3-(2-methylpropyl)-8-(quinolin-6-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{2-[1-(6-fluoro-4-hydroxyquinoline-3-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
3-[(2,8-dimethylquinolin-4-yl)formamido]-N-(1,3-thiazol-2-yl)propanamide
1-{6-[4-(methoxymethyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}azepane
{4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1,4-oxazepan-6-yl}methanol
7-(pyridin-3-ylmethyl)-2-(thian-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[2-(4-phenyl-1H-imidazol-5-yl)phenoxy]ethan-1-ol
4-methyl-2-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
methyl 4-({[1-(pyrimidin-2-yl)piperidin-3-yl]amino}methyl)benzoate
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-methanesulfonyl-N-(pyridin-3-ylmethyl)acetamide
4-[4-({[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]-2-methylbut-3-yn-2-ol
2-(2,2-diphenylethyl)-4-[(4-methyl-1H-imidazol-5-yl)methyl]morpholine
2-hydroxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-5-(1H-pyrrol-1-yl)benzamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
6-{[(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)amino]methyl}-1,4-oxazepan-6-ol
N-methyl-N-(1-{1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}-2-phenylethyl)thiophene-3-carboxamide
6-(benzyloxy)-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
2-[3-(pyridine-2-carbonyl)piperidin-1-yl]-4-(3,3,3-trifluoropropyl)pyrimidine
3-{2-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-(cyclohex-1-en-1-ylmethyl)-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
5-acetyl-N-butyl-N-(furan-2-ylmethyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
ethyl 4-(6-methyl-3-{[(propan-2-yl)amino]methyl}quinolin-2-yl)piperazine-1-carboxylate
2-(morpholin-4-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-2-(pyridin-3-yl)acetamide
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}furan-3-carboxamide
6-{[3-(4-phenylbenzoyl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-cyclobutyl-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
2-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]thiophene-3-sulfonamide
methyl 5-[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-5-oxopentanoate