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ethyl 1-(dimethylsulfamoyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
N-(2-methoxyethyl)-N-[(5-methylthiophen-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-[1-(2,2-dimethylpropyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
N-(1-cycloheptylpiperidin-3-yl)-2-methoxyacetamide
N-(5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-2-methylphenyl)butanamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
1-[2-(dimethylamino)-4-{[(5-ethylpyridin-2-yl)methyl](methyl)amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-cyclopentyl-4-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
3-oxo-N-phenyl-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-(cyclohexylmethyl)-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
5-oxo-1-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}pyrrolidine-3-carboxylic acid
(1R,5R)-6-(1H-indol-5-ylmethyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-3-{4-[3-(morpholin-4-yl)-3-oxopropyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-(2-methoxyethyl)-9-[(2-propoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-(2-hydroxyphenoxy)ethan-1-one
{1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
5-[(3-methoxyphenyl)methyl]-3-methyl-5-(piperidin-4-yl)imidazolidine-2,4-dione
methyl({[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
6-methyl-4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amine
4,5-dimethyl-2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-1,3-benzodiazole
(3S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-[methyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]pyrrolidin-3-ol
methyl 1-(2-methoxyethyl)-3-(3-phenylpropanamido)-5-[(thiophen-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(4S)-1-(2-chloro-6-fluoro-3-methylbenzoyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
4-[3-(3-methoxypropyl)piperidine-1-carbonyl]-6-methylquinoline
4-methoxy-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-phenylpiperidine
N-{4-[2-(hydroxymethyl)phenyl]-2-methylphenyl}pyridine-3-carboxamide
(3S,4S)-4-(4-fluorophenyl)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-ol
1-(3,5-dimethylphenyl)-4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
3-{[(3-{2-azabicyclo[2.2.1]hept-5-en-2-yl}propyl)amino]methyl}-N,8-dimethyl-N-(thiophen-2-ylmethyl)quinolin-2-amine
N-{[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
1-methyl-2-(morpholin-4-yl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
4-{1-[6-(1H-pyrazol-4-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
2-{5-[(3S)-3-ethylmorpholine-4-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
6-methyl-3-[(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-4H-chromen-4-one
4-(cyclopropylmethyl)-1-(3-methylbenzoyl)-1,4-diazepan-5-one
1-{5-[(ethylamino)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-N-(thiophen-2-ylmethyl)piperidine-4-carboxamide
4-[6-(3-methyl-1H-pyrazol-5-yl)pyridine-3-carbonyl]morpholine
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methylpyrrolidine-3-carboxamide
(1R,5R)-N,N-dimethyl-6-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(1H-1,2,4-triazol-3-yl)benzamide
2-{1-cyclohexyl-5-[2-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-oxo-6-({4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}methyl)-1,2-dihydropyridine-3-carboxamide
6-methyl-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-2-(pyridin-3-yl)pyrimidin-4-amine
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(4-phenoxyphenyl)methyl]amine
2-ethyl-6-(4-ethyl-5-methylthiophene-3-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
4-{1-cyclohexyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}benzonitrile
(benzylsulfamoyl)[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]amine
N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine