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4-[4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]quinazoline
1-[5-(3-methoxyphenyl)furan-2-carbonyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
1-(cyclopropylmethyl)-5-({[4-(pyrrolidine-1-carbonyl)phenyl]methyl}amino)azepan-2-one
[7-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
methyl (2S,4S)-4-(4-fluorobenzamido)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
({2-[4-(3-chlorophenyl)piperazin-1-yl]-7-fluoroquinolin-3-yl}methyl)[(3,4-dimethoxyphenyl)methyl]amine
2-[5-(5-fluoro-1-methyl-1H-indol-2-yl)-3-methyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
2-[2,4-dioxo-1-(2-phenylethyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
4-(1-hydroxybutan-2-yl)-11-methyl-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(naphthalen-1-ylmethyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-5-methoxyfuran-2-carboxamide
N-(5-methyl-1,2-oxazol-3-yl)-N'-[(3-methylphenyl)(thiophen-2-yl)methyl]ethanediamide
(2,3-dihydro-1-benzofuran-2-ylmethyl)({[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
2-amino-6-cyclopropanecarbonyl-4-(quinolin-5-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3R,4S)-1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-3,4-dimethylpiperidin-4-ol
methyl[(2E)-2-methylbut-2-en-1-yl][(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
2-(4-{[4-(2,2-dimethylpropyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
4-[(2-ethylpyrimidin-5-yl)methyl]-2-[(3-fluorophenyl)methyl]morpholine
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropane-1-carboxamide
1-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]urea
3-{1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidin-3-yl}benzoic acid
N-{imidazo[1,2-a]pyrazin-3-ylmethyl}-3-phenoxypropanamide
7-(2-methylphenyl)-4-(pyrrolidine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(3-methylphenoxy)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}azetidine
N-[(4-hydroxyazepan-4-yl)methyl]-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-sulfonamide
[(3R,4R)-1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-{2-oxo-2-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethyl}-1,2-dihydropyrimidin-2-one
(4aS,7aR)-1-[(2,6-dichlorophenyl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}oxolane-2-carboxamide
1-({3-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-indole
[(2-methoxyphenyl)methyl][(3-phenyloxolan-3-yl)methyl](pyridin-3-ylmethyl)amine
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
(1S,9S)-11-[(8-methoxy-2H-chromen-3-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
7-methyl-2-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
(5-{1-[2-(ethylsulfanyl)ethyl]-4-phenyl-1H-imidazol-5-yl}furan-2-yl)methanol
4-({3-hydroxy-1-[(3-methylphenyl)methyl]-2-oxopiperidin-3-yl}methyl)-3,3-dimethylpiperazin-2-one
4-(2-cyclopropylpyrimidine-5-carbonyl)-2-(trifluoromethyl)morpholine
(2S,3R)-2-amino-1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-hydroxybutan-1-one
1-(carbamoylmethyl)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]piperidine-4-carboxamide
1-(4-methyl-1H-imidazole-5-carbonyl)-3-(1H-pyrazol-5-yl)piperidine
4-methoxy-6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
N-phenyl-6-[(2E)-3-(pyridin-3-yl)prop-2-enoyl]-6-azaspiro[2.5]octane-1-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
1-[(3-chlorophenyl)methyl]-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]thieno[2,3-d]pyrimidin-4-amine
N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
4-[2-chloro-5-(trifluoromethoxy)phenyl]pyridin-3-amine
N-(3,5-dimethoxyphenyl)-3-[1-(1H-indole-3-carbonyl)piperidin-3-yl]propanamide