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3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}({[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl})amine
4-(5-methoxypyridin-3-yl)-6-(4-methyl-1H-pyrazol-1-yl)pyrimidine
2,6-dimethyl-7-(4-phenyl-1H-imidazol-5-yl)heptan-2-ol
2-{4-[(3,5-dimethyl-1H-indol-2-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-3-methoxy-2,2-dimethylpropanamide
ethyl 1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[benzyl(methyl)amino]-3-{4-[({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amino)methyl]phenoxy}propan-2-ol
1-(oxan-2-ylmethyl)-1,2-dihydroquinoxalin-2-one
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(3-methoxyphenyl)propan-1-one
1-[2-(pyridin-2-yl)-4-[(thiophen-2-ylmethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
9-[(dimethyl-1,3-thiazol-5-yl)methyl]-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
7-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-sulfonyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazine
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
6-{3-[(1-methylpiperidin-4-yl)oxy]propyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-cyclopentyl-N-[(2,5-dimethoxyphenyl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
2-{4-[1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperazin-1-yl}phenol
[(2S)-1-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidin-2-yl]methanol
1-(1-methyl-1H-pyrrole-2-carbonyl)-2-(2-phenylethyl)piperidine
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-[(5-methylpyrazin-2-yl)methyl]propanamide
1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(pyridin-4-yl)propan-1-one
3-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-N-[2-(1H-pyrazol-1-yl)ethyl]benzene-1-sulfonamide
8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(dimethylamino)ethyl]-3-{2-[4-(2,4-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}-3-(2-fluorophenyl)pyrrolidine-2,5-dione
2-[4-(5-fluoropyridin-2-yl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
N-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-2-(methylamino)acetamide
4-(5-methyl-1,3,4-oxadiazol-2-yl)-N,N-diphenylpiperazine-1-carboxamide
N-[(2R,3R)-1'-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
4-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-(propan-2-yl)-1H-pyrazole
1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
(4-{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-oxazepan-6-yl)methanol
8-[2-(1H-imidazol-1-yl)acetyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(4aR,7aS)-1-methyl-4-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-6-(4-ethoxybenzoyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(3-fluorophenoxymethyl)-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine
4-[3-(4-fluorophenoxy)azetidine-1-carbonyl]-2,7,8-trimethylquinoline
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-N-cyclopentyl-4-oxobutanamide
2-methoxy-4-[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]pyridine
1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-methoxy-N-[2-(3-phenylprop-2-ynoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
2-{4-[2-(dimethylamino)ethoxy]piperidin-1-yl}-2-(6-methoxynaphthalen-2-yl)acetic acid
2-(3-fluoropropyl)-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
(1R,3S,5S)-3-(4-methoxyphenyl)-8-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-8-azabicyclo[3.2.1]octane
2-(ethylamino)-N,4-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,3-thiazole-5-carboxamide
2,5-dioxo-6-[2-(3-phenylpiperidin-1-yl)ethyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-2-one
N-[2-(azepan-1-yl)ethyl]-N-(propan-2-yl)-1,2,3-thiadiazole-4-carboxamide
(1R,5R)-6-benzyl-3-(pyrrolidine-1-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane