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N-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}methyl)acetamide
N-[2-(dimethylamino)ethyl]-3,5,7-trimethyl-N-(oxolan-2-ylmethyl)-1H-indole-2-carboxamide
(2S,4S)-4-{[(3,4-difluorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
({4-[1-(1H-imidazol-2-ylmethyl)piperidin-2-yl]phenyl}methyl)dimethylamine
ethyl 4-(2-phenylethyl)-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-4-carboxylate
1-(1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)piperidin-3-ol
2-(2,4-dimethoxy-3-methylphenyl)-6-fluoro-1H-1,3-benzodiazole
3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
4-(2,6-dimethylphenyl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenoxy}acetamide
N-butyl-N-methyl-3-{[(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
3-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-9-methoxy-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
(3R,5R)-1-benzyl-N-(2-methylpropyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
5-[2-(methylsulfanyl)phenoxymethyl]-3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,2-oxazole
N-methyl-N-[2-(oxan-4-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
2-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-(ethylamino)-N-[(4-phenylphenyl)methyl]pyrimidine-5-carboxamide
(2S)-2-[(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)formamido]-3-(4-hydroxyphenyl)propanamide
N-[4-({4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepan-1-yl}methyl)phenyl]acetamide
N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
2-{[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}-2-[4-(methylsulfanyl)phenyl]acetic acid
5-[1-(2,6-difluorobenzoyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
3-(4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
3-(2-{4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
(1S,5R)-3-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(5-{1-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-imidazol-2-yl}thiophen-3-yl)prop-2-yn-1-ol
ethyl 1-(1H-indazol-7-yl)-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
1-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
N,N-diethyl-1-({1-[(2Z)-3-(3-fluorophenyl)prop-2-enoyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
N-(1-{7-[(3-ethoxy-2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)propanamide
2-(2,4-difluorophenyl)-5-(4-methoxy-4-methylpentan-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-{2-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
4-{1-[(2,4-dimethoxyphenyl)methyl]piperidin-4-yl}-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
N-(1-{7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
6-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-[3-methoxy-5-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
(3R,4R)-1-[(2,5-dimethoxyphenyl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
N-(1-cyclopentyl-1H-pyrazol-5-yl)-4-(2-methoxyphenoxy)piperidine-1-carboxamide
N-methyl-4-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}methyl)benzene-1-sulfonamide
N-benzyl-1-(2-hydroxyethyl)-5-[(2E)-3-phenylprop-2-en-1-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-benzyl-3-(2-methyl-1,3-thiazol-4-yl)-5-[(oxolan-2-ylmethoxy)methyl]-1H-1,2,4-triazole
N-(1,3-benzoxazol-2-ylmethyl)-2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
8-(azepane-1-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1R,5R)-3-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[1-(pyridin-4-yl)propyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-(1,5-dimethyl-1H-indazole-3-carbonyl)-3-[(dimethylamino)methyl]pyrrolidin-3-ol
8-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
7-[1-(4-chlorophenyl)cyclobutanecarbonyl]-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-methanesulfonamido-N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}propanamide