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4-[3-(benzyloxy)azetidin-1-yl]-2,5,6-trimethylpyrimidine
1-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]azetidin-3-yl}-2-methylpiperidine
(3aR,6aR)-N-ethyl-2-(2-methoxyacetyl)-N-(pyridin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-(1-{7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
7-chloro-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-9-oxo-9H-fluorene-1-carboxamide
9-(5-ethyl-2-methylpyrimidin-4-yl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-benzyl-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-one
N-[1-(2,5-difluorophenyl)cyclopropyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-methyl-1,4-dihydroquinolin-4-one
N-[5-(2-methoxypyridin-3-yl)pyridin-2-yl]methanesulfonamide
4-[(1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]benzoic acid
2-(1H-indol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(2-{[(2-methoxynaphthalen-1-yl)methyl]amino}ethyl)-N-(2-methylphenyl)-1H-1,2,3-triazole-4-carboxamide
1-[1-(3-methoxybenzoyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
4-{[6-(dimethylamino)pyridin-3-yl]methyl}-1,4-oxazepan-6-ol
2-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-ethyl-N-methylacetamide
2-(3-methoxyphenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
ethyl 4-{1-[2-(3-chloro-4-methoxyphenyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carbonyl}piperazine-1-carboxylate
[(2-methoxyphenyl)methyl][(2-methyl-1H-imidazol-4-yl)methyl](pyridin-3-ylmethyl)amine
{4-benzyl-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methanol
4-hydroxy-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-1,3-thiazole-5-carboxamide
3-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-[4-(oxan-2-ylmethoxy)phenyl]urea
5-tert-butyl-3-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}-1H-pyrazole
1-[(2-methoxyphenyl)methyl]-N3-(3-methylbutyl)-4-oxo-N5-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(1S,5R)-3-cyclobutanecarbonyl-N-(2-fluorophenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
N-(2-methanesulfonylethyl)-4-methyl-7-(methylsulfanyl)quinolin-2-amine
5-methyl-N-[(5-methylpyrazin-2-yl)methyl]-3-phenyl-1,2-oxazole-4-carboxamide
1-(1-cyclobutanecarbonylpiperidin-4-yl)-N-(2-phenylethyl)piperidine-3-carboxamide
[1-(2,1,3-benzothiadiazole-4-sulfonyl)-3-benzylpiperidin-3-yl]methanol
(1S,5R)-3-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1-{[3-(furan-2-yl)phenyl]methyl}-4-[(4-methoxyphenyl)methyl]piperidin-4-yl)methanol
3-(2H-1,3-benzodioxol-5-yl)-5-(thiolan-3-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
1-[2-(dimethylamino)ethyl]-6-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
2-{4-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]piperidin-1-yl}acetamide
3-benzoyl-1-(2,3-difluorobenzoyl)piperidine
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-[2-(2-methoxyphenyl)ethyl]-6-(3-phenylbutyl)-6-azaspiro[2.5]octane-1-carboxamide
6-fluoro-2-(thiomorpholin-4-ylmethyl)quinolin-4-ol
N'1-{4-[(3-methoxyphenyl)carbamoyl]phenyl}cyclopropane-1,1-dicarboxamide
[3-(1H-imidazol-1-yl)propyl]({[2-(propan-2-yl)pyrimidin-4-yl]methyl})(pyridin-3-ylmethyl)amine
2-ethoxy-6-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenol
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,2-oxazole-3-carboxamide
2-(4-ethoxyphenyl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
8-fluoro-2-({[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amino}methyl)quinolin-4-ol
2-{1-[(3-methoxyphenyl)methyl]-4-{[4-(trifluoromethyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N-[2-(pyridin-2-yl)ethyl]pyrimidin-2-amine
methyl (1R,3S,3aR,6aS)-1-ethyl-3-[4-(1H-imidazol-1-yl)phenyl]-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate