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3,3,3-trifluoro-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]propanamide
3-{2-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}piperidin-2-one
ethyl 4-[(4-methoxyphenyl)methyl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine-4-carboxylate
N-[(3R,4S)-4-cyclopropyl-1-[(2-methoxyphenyl)methyl]pyrrolidin-3-yl]oxane-4-carboxamide
2-methyl-6-(2-phenoxyethyl)-[1,2,4]triazolo[1,5-a]pyridine
1-[1-ethyl-5-(2-methylbenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
(3R,9aR)-8-(4-methylbenzenesulfonyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[3-(benzyloxy)propyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5-propyl-1,3,4-oxadiazol-2-amine
4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-(2-methoxyphenyl)-2,2-dimethylpiperazine
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
N3-methyl-N3-(2-methylpropyl)-4-oxo-N5-(3-phenylpropyl)-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-4-phenylpiperidin-4-ol
methyl 3-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[(3R,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-methyl-2-(1-methyl-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-4-yl)-N-(oxan-2-ylmethyl)acetamide
7-[3-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[3-(methylsulfanyl)propyl]-1,2-oxazole-3-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(naphthalen-2-ylmethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(1R,3S,5S)-8-[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-8-azabicyclo[3.2.1]octan-3-ol
2-benzyl-8-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-2,8-diazaspiro[4.5]decan-3-one
3-ethyl-N,5-dimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1,2-oxazole-4-carboxamide
ethyl 3-({3-[(furan-2-ylformamido)methyl]piperidine-1-carbonyl}amino)propanoate
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyrimidin-4-ylmethyl)amine
1-cyclopropyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-oxopyrrolidine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-ethyl-N,6-dimethylpyrimidin-4-amine
5-ethyl-2-methyl-4-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}pyrimidine
1-[2-(cyclohex-1-en-1-yl)ethyl]-1-(cyclopropylmethyl)-3-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
N-(dicyclopropylmethyl)-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-{4-[(methylsulfanyl)methyl]piperidin-1-yl}-4-(trifluoromethyl)pyrimidine
1-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-hydroxypropan-1-one
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]acetamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
[(1-butyl-1H-1,2,4-triazol-5-yl)methyl][(2-fluorophenyl)methyl]methylamine
3-hydroxy-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-4-methylbenzamide
1-[(2-chlorophenyl)methyl]-N-methyl-N-[3-(morpholin-4-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
9-(cyclopropylmethyl)-4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
6-methyl-1-{3-oxo-3-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}-1,2-dihydropyridin-2-one
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pentane-1,2-dione
N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
(1R)-1-[(4-methoxyphenyl)methyl]-2-(1H-1,2,3-triazole-5-carbonyl)-1,2,3,4,5,6,7,8-octahydroisoquinoline
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(5-methylthiophen-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2-fluoropyridin-3-yl)-3-methyl-3-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]urea
9-methoxy-7-(6-methoxypyridin-2-yl)-4-(propan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[4-(4-methoxyphenyl)-5-methyl-1H-imidazol-2-yl]-1-[(4-methylphenyl)methyl]pyrrolidin-2-one
4-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-1λ6-thiane-1,1-dione
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-5-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(3S)-3-ethylmorpholin-4-yl]-3-(pyridin-2-yl)propan-1-one
N-[(3R,4S)-1-(carbamoylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
3,3,3-trifluoro-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one