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1-ethyl-4-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
2-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-(4-benzoylpiperazin-1-yl)ethan-1-one
N-[2-(3-chlorophenyl)ethyl]-4-methylpyrimidine-5-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(6-hydroxypyrimidin-4-yl)ethyl]acetamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]propan-1-one
({[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]methyl}sulfamoyl)dimethylamine
4-[2-(1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-2-yl)ethyl]phenol
3-cyclopropaneamido-4-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
5-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-(2-methylpropyl)-1H-imidazole
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(morpholin-3-yl)acetamide
N-[2-(dimethylamino)ethyl]-1-methyl-N-[(3-methylthiophen-2-yl)methyl]-1H-1,2,3-benzotriazole-5-carboxamide
N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-1,2,3,4-tetrahydroquinoline-8-carboxamide
9-(but-3-yn-1-yloxy)-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-ethyl-3-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(3-hydroxy-3-methylbutyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]benzamide
methyl 4-methyl-3-({[2-(pyrrolidine-1-sulfonyl)ethyl]carbamoyl}amino)benzoate
N-{1-[1-(2-methoxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
(3S,4R)-4-phenyl-1-[2-(pyridin-3-yl)acetyl]pyrrolidine-3-carboxylic acid
5-ethyl-1'-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(2-methylprop-2-en-1-yl)benzamide
4-fluoro-N-{2-[1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]ethyl}benzamide
N-[2-(dimethylamino)ethyl]-1-[1-(2-fluorobenzoyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
6-[(2-hydroxy-3-methoxyphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-6-azaspiro[2.5]octane-1-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-methyl-N-(oxan-4-yl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methoxy-2,2-dimethylpropan-1-one
N-[2-(tert-butylsulfanyl)ethyl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
9-(5-chloro-2-methylpyrimidine-4-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
4-{4-[2-(2-methyl-5-oxopyrrolidin-1-yl)acetyl]piperazin-1-yl}benzonitrile
2-{1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl}-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
2-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)-N,N-dimethylacetamide
1-[cyclohexyl(methyl)amino]-3-[4-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]propan-2-ol
4-fluoro-2-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}phenol
1-(3-methylbut-2-en-1-yl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(trifluoromethyl)pyrimidin-2-amine
5-phenoxy-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]furan-2-carboxamide
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(2-methoxyphenyl)methyl]pyrrolidin-3-yl]methanol
2-{2-oxa-7-azaspiro[4.5]decan-7-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
N-cyclopropyl-4-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]piperazine-2-carboxamide
methyl (1R,3S,3aR,6aS)-5-ethyl-4,6-dioxo-3-[2-(trifluoromethyl)phenyl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-5-(propan-2-yl)pyrimidin-4-amine
[(2S,6S)-4-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
ethyl 4-[(3-methoxyphenyl)methyl]-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine-4-carboxylate
N-[2-(1H-imidazol-4-yl)ethyl]-2-(1-methylpiperidin-4-yl)acetamide
N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
methyl (2S,4R)-4-(2,3-dimethyl-1H-indole-7-amido)-1-[(4-ethylphenyl)methyl]pyrrolidine-2-carboxylate
N-methyl-N-(1-methylpiperidin-4-yl)-2-phenylimidazo[1,2-a]pyridine-6-carboxamide