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N-ethyl-2-(1-ethyl-1H-pyrazol-4-yl)-7-methyl-N-(pyridin-4-ylmethyl)quinoline-4-carboxamide
N-methyl-N-[1-(thiophen-2-yl)ethyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(1H-1,3-benzodiazol-2-ylmethyl)(methyl)[(5-methyl-1,2-oxazol-3-yl)methyl]amine
N-methyl-2-{4-[2-(phenylsulfanyl)acetamido]-1H-pyrazol-1-yl}-N-(quinoxalin-6-ylmethyl)acetamide
N-{[4-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)cyclohexanecarboxamide
5-methyl-1-(4-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}phenyl)-1H-1,2,3,4-tetrazole
1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-N-[1-(thiophen-3-yl)propan-2-yl]piperidin-4-amine
1-{4-[2-(cyclohexylmethyl)morpholin-4-yl]-4-oxobutyl}piperidin-2-one
4-(4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)quinazoline
3-(2-methylpropyl)-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1,2-oxazole-5-carboxamide
5-{1-[3-(diethylamino)propanoyl]piperidin-4-yl}-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
7-(1,3-benzothiazol-2-yl)-4-(furan-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-methoxy-7-(3-methoxyphenyl)-4-[(4-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-[5-(3,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-2-methylheptan-2-ol
2-amino-6-(6-chloro-1H-1,3-benzodiazol-2-yl)-4-(1,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
{2,4,6-trimethyl-3-[5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazol-2-yl]phenyl}methanol
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
2-{5-cyclopropyl-4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(2-fluorophenyl)pyrimidine
2-(4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholin-2-yl)ethan-1-amine
N-[3-(3,4-diethoxyphenyl)propyl]-2-hydroxyacetamide
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-[4-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-(1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide
N-(2-{7-[(2-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
N-cyclopropyl-4-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]pyridine-2-carboxamide
4-{3-[(4-methyl-3-phenylpiperazin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}morpholine
2-butanoyl-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
methyl 3-[(2-cyclopentylacetamido)methyl]-5-(2,3-dihydro-1,4-benzodioxine-6-sulfonamido)benzoate
(3S,4S)-3-[(1-ethylpiperidin-4-yl)(methyl)amino]-4-hydroxy-1λ6-thiolane-1,1-dione
7-[ethoxy(phenyl)methyl]-4-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
[2-(1H-imidazol-1-yl)ethyl](methyl){[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amine
1-[(2-methyl-1H-imidazol-4-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
4-phenyl-3-{1-[1-(propan-2-yl)piperidin-4-yl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(5-{[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}furan-2-yl)methanol
2-(3-hydroxypropyl)-8-[(2-methoxy-3,5-dimethylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-(2,4-dioxoimidazolidin-1-yl)-N-[(2-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)benzamide
1-ethyl-N-methyl-3-(2-methylpropyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
4-[(1-cyclohexyl-3-phenyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-2-one
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1-methoxy-2-methylpropan-2-yl)propanamide
N-methyl-N-propyl-2-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
4-[2-(ethylamino)pyrimidine-5-carbonyl]-1-[(4-fluorophenyl)methyl]piperazin-2-one
2-ethyl-4-(2-methyl-1,3-thiazole-5-carbonyl)-1-(propan-2-yl)piperazine
1-{2-[2-(3-fluorophenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]piperidine-4-carboxamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]but-3-enamide
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl){[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}amine
1-(3-methyl-1H-pyrazole-4-carbonyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-2-ylmethyl)piperidine
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-2-(thiophen-2-yl)-1,3-thiazole
2-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[3-(pyridin-3-yl)propyl]propanamide
5-chloro-15-methyl-13-oxo-N-(oxolan-2-ylmethyl)-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide