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5-(1-{2-[4-(methylsulfanyl)phenyl]acetyl}piperidin-4-yl)-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
5-{3-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-oxopropyl}-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
3-[(3R,4S)-1-(6-aminopyrimidin-4-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-(1-methyl-1H-indole-4-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1,8-naphthyridine
3-chloro-4-fluoro-N-[1-(pyrimidin-4-yl)ethyl]-1-benzothiophene-2-carboxamide
1,3-dimethyl-4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-1H-pyrazolo[3,4-d]pyrimidine
6-(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)-2-methylpyrimidin-4-ol
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
1-(4-chlorophenyl)-N-({1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
N-(oxan-3-ylmethyl)-3-[(pyridin-4-ylmethyl)sulfamoyl]benzamide
N-[(7-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
6-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N,2-dimethylquinoline-4-carboxamide
N-[1-({[2-(cyclohex-1-en-1-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]benzamide
N3-tert-butyl-1-cyclohexyl-4-oxo-N5-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-{[3-(2-methylpropyl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R,6R)-4-[4-(1H-imidazol-1-yl)benzoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1,3-thiazol-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N,N-dimethylpyridin-2-amine
N-[(1R,3R)-3-aminocyclopentyl]-2-(3-butanoyl-1H-indol-1-yl)acetamide
4,6-dimethyl-2-(quinolin-3-yl)pyridine-3-carboxamide
N-(2-fluoroethyl)-3-[(3-methoxypropyl)(methyl)sulfamoyl]benzamide
N-cyclopentyl-4-(4-{[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)benzamide
5-methanesulfonyl-N-[(1-methylpiperidin-4-yl)methyl]-4-(piperidin-3-yl)pyrimidin-2-amine
N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,3-oxazole-4-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-(morpholine-4-carbonyl)pyrrolidin-3-yl]acetamide
N-cyclohexyl-2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzamide
2,6-dimethyl-4-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenol
diethyl[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)sulfamoyl]amine
(2S,4R)-N,N-diethyl-4-[2-(3-fluoro-4-hydroxyphenyl)acetamido]-1-methylpyrrolidine-2-carboxamide
2-[2-(carbamoylmethoxy)-5-methylphenyl]benzamide
2-ethyl-7-methoxy-4-[(2-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[2-(trifluoromethyl)phenyl]methyl}amine
3-cyclohexyl-N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-1H-pyrazole-4-carboxamide
2-{[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{[1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxy}quinoxaline
1-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
2-phenoxy-N-[(7-{[4-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-4-(pyridin-4-yl)pyrimidin-2-amine
(4aR,7aS)-1-(cyclopropylmethyl)-4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 6-{[benzyl(methyl)amino]methyl}-3-(1,3-dimethyl-1H-pyrazole-5-amido)thieno[2,3-b]pyridine-2-carboxylate
N-(3-benzyl-1H-1,2,4-triazol-5-yl)-4-(1,3,5-triazin-2-yl)piperazine-1-carboxamide
1-(4-ethoxyphenyl)-3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
N-[1-(3-phenylpropyl)piperidin-3-yl]-2-(pyrimidin-2-ylsulfanyl)acetamide
(2S,4S)-4-[3-(difluoromethoxy)benzamido]-N,N-diethyl-1-methylpyrrolidine-2-carboxamide
N4-methyl-N4-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}acetamide
3-(4-methyl-1,3-thiazol-5-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
4-{[2-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
(2S,4S)-4-(3,4-difluorobenzamido)-N-ethyl-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide