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N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(2-hydroxyethyl)piperidin-4-yl]methyl}acetamide
1-methyl-N-(3-methylbutyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-methyl-N-[(1-methylpiperidin-3-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
(3S,5R)-1-(4,6-dimethylpyrimidin-2-yl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]morpholine-2-carboxamide
2-amino-4-{2-[2-(morpholin-4-yl)ethoxy]phenyl}-5H,6H,7H,8H,9H-cyclohepta[b]pyridine-3-carbonitrile
N-methyl-7-oxo-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
1-{3-oxo-3-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]propyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(2R,3R)-2-methoxy-1'-(quinolin-8-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
3-[1-cyclohexyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-2-(methylsulfanyl)pyridine
7-[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[3-({[3-(2-ethyl-1H-imidazol-1-yl)propyl]carbamoyl}amino)-4-methoxyphenyl]acetamide
N-{[1-(1-methyl-2-oxo-1,2-dihydroquinoline-4-carbonyl)piperidin-3-yl]methyl}furan-2-carboxamide
2-[2-oxo-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]acetamide
2-(1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-1H-imidazol-2-yl)-1-methyl-1H-imidazole
7-(2-methoxypyridine-3-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(5-ethylpyridin-2-yl)methyl]-4-(thian-4-yl)piperazine
2-(4-propylpyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
6-(3-chlorophenyl)-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)pyridine-3-carboxamide
3-methyl-1-(1-{6-[(pyridin-4-ylmethyl)amino]pyridine-3-carbonyl}piperidin-3-yl)butan-1-one
5-(4-fluorophenyl)-2-methyl-4-{1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}pyrimidine
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-(oxane-4-carbonyl)piperidine
2-[2-(5-butyl-4-phenyl-1H-imidazol-1-yl)propyl]pyrazine
1-{1-[(4,6-dimethylpyrimidin-2-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
2-[5-(2-methoxyethyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
5-{3-[(4-fluorophenyl)amino]piperidine-1-carbonyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
methyl (2S,4R)-4-[2-chloro-5-(1H-pyrazol-1-yl)benzamido]-1-methylpyrrolidine-2-carboxylate
5-(cyclopropylmethyl)-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(3-fluoropyridin-4-yl)piperidine-4-carboxylic acid
1-methyl-4-{5-[1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]thiophene-2-carbonyl}-1,4-diazepane
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-(3-methyl-1,2-oxazol-5-yl)-1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-N-[(1-ethylpyrrolidin-2-yl)methyl]acetamide
N-[2-(furan-2-yl)ethyl]-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
4-[(3-acetamidopyrrolidin-1-yl)methyl]-N-(3-ethylphenyl)benzamide
(1R,3S,5S)-8-[(2-butoxy-3-methoxyphenyl)methyl]-8-azabicyclo[3.2.1]octan-3-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-N-[3-(dimethylamino)-2,2-dimethylpropyl]-5-methoxybenzamide
(3R,4S)-4-cyclopropyl-1-(6-methylpyridazin-3-yl)pyrrolidin-3-amine
(5S,9aS,9bS)-5-[(E)-2-(furan-2-yl)ethenyl]-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(4aS,7aR)-1-[(2-ethylphenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-methyl-1,3-thiazol-4-yl)-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]acetamide
4-(2-phenoxyethyl)-1,3λ6,4-oxathiazinane-3,3-dione
N-(adamantan-1-yl)-2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}acetamide
2-ethyl-5-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-4-methyl-1,3-oxazole
2-[(1S,5R)-6-(2-acetylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
6-methyl-4-oxo-1-(oxolan-2-ylmethyl)-2-(2-phenylethyl)-N-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
2-{1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-2-yl}pyridine