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4-(5-acetylthiophene-3-carbonyl)-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
(4aS,7aR)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1H-1,2,3-triazole-5-carboxamide
2-(3-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-1H-indol-1-yl)acetamide
4-(4-chlorophenyl)-N-(2-hydroxy-1-phenylethyl)butanamide
N-ethyl-N-methyl-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
2-chloro-4-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-6-methoxyphenol
2-cyclobutanecarbonyl-8-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}-6-(pyrrolidine-1-carbonyl)pyrazine
1-ethyl-N-[(2-fluorophenyl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-ethyl-N,4-dimethyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-1H-pyrazole-5-carboxamide
5-(1,2-dihydroacenaphthylen-5-yl)-1,3-dimethyl-1H,4H-pyrazolo[3,4-d]imidazole
4-hydroxy-2-methyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}pyrimidine-5-carboxamide
4-{[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}benzene-1-sulfonamide
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[4-(2-phenoxyethyl)piperazin-1-yl]propan-1-one
N-methyl-4-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]-1,3-thiazol-2-amine
4-[(2-aminopyrimidin-5-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(methylamino)-N-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)pyrimidine-5-carboxamide
2-amino-6-(2,2-dimethylcyclopropyl)-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-5-methylpyridine-3-carbonitrile
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
2-(4-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}phenyl)ethan-1-amine
9-[(5-propylfuran-2-yl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{2-[1-(1H-indole-6-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
methyl({[2-(2-methylphenyl)pyrimidin-5-yl]methyl})(oxan-2-ylmethyl)amine
1-(4-{[(3R,4S)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
2-{4-chloro-2-[1-(furan-2-ylmethyl)-1H-imidazol-2-yl]phenoxy}acetamide
N-[(2R,3R)-2-(pyridin-2-ylmethoxy)-1'-[3-(thiophen-2-yl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
1-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(pyrrolidin-1-yl)propan-1-one
methyl 1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)azetidine-3-carboxylate
1-(2-phenylethyl)-3-(propan-2-yl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[2-methyl-2-(morpholin-4-yl)propyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(3R,4R)-4-(azepan-1-yl)-1-[1-(3-methylphenyl)piperidin-4-yl]piperidin-3-ol
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(pyrrolidine-1-carbonyl)piperidine
N-(5-chloro-2-methoxyphenyl)-3-[1-(cyclopropanesulfonyl)piperidin-3-yl]propanamide
methyl 5-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amine
2-[(3S,4R)-3-acetamido-4-(4-methoxyphenyl)pyrrolidin-1-yl]-N-(furan-2-ylmethyl)acetamide
2-{1-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]-1H-imidazol-2-yl}benzoic acid
N-methyl-N-[(4-methylphenyl)methyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
(4aS,8aR)-6-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
(3R,9R)-11-(naphthalene-1-carbonyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
2-cyclopentyl-8-(1-propyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(4-hydroxyphenyl)ethyl]-4-(piperidin-1-yl)butanamide
1-{[(2S,4S)-1-(1,3-benzothiazole-6-carbonyl)-4-fluoropyrrolidin-2-yl]methyl}-3,3-dimethylurea
ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}){[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
4-[3-(4-hydroxyphenyl)benzoyl]-N,N-dimethylpiperazine-1-carboxamide
{5-methyl-7-[3-(pyrrolidin-1-yl)pyrazin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
N,3,5,7-tetramethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1H-indole-2-carboxamide
1-{2-[1-(2,4-difluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}-4-methylpiperazine