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(4aS,7aR)-6,6-dioxo-N-phenyl-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-4-oxo-N-(1,3,4-thiadiazol-2-yl)butanamide
4-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-[3-(pyridin-4-yl)propanoyl]-1,4-diazepan-2-one
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1H-pyrazol-4-yl)propan-1-one
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-[(2R)-oxolane-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(3-{2-[(2-methoxyethyl)sulfanyl]-5-(3-methoxyphenyl)pyrimidin-4-yl}piperidin-1-yl)methyl]-1H-1,3-benzodiazole
(2S,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
1-[2-(1-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
2-[2-methyl-2-(thiophen-2-ylformamido)propanamido]-4-(methylsulfanyl)butanoic acid
(1S,5R)-N-(3-chlorophenyl)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]acetamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-1-benzofuran-3-carboxamide
5-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-(4-ethyl-1H-pyrazol-5-yl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
N-[2-(1H-imidazol-4-yl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
3,5-dimethyl-1-phenyl-4-({3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-1H-pyrazole
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-(4-methoxyphenyl)-5-methyl-1H-pyrazole
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-amino-4-{[1-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}quinazoline-6-carboxylic acid
N-[2-(dimethylamino)ethyl]-4-(3-methylphenyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
9-[(2E)-3-phenylprop-2-en-1-yl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-{[(3-chlorophenyl)methyl]sulfamoyl}-6-(4-methylpentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-(thiophen-2-yl)propan-1-one
2-(4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
(3aR,6aS)-N-[4-ethoxy-3-(trifluoromethyl)phenyl]-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
N,N-dimethyl-2-{[2-(1-methylpiperidin-2-yl)acetamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-3-[4-(2-methylpropoxy)phenyl]-1H-pyrazole
2-({2-methyl-4-[(3-methylphenyl)methyl]-3-oxopiperazin-1-yl}methyl)pyridine-3-carboxylic acid
1-cyclohexyl-N3-(1,2-diphenylethyl)-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-[(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-2-methoxybenzoic acid
N-(2-methoxyethyl)-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)urea
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
1-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}-4-[3-(trifluoromethyl)phenyl]piperazine
N-methyl-4-(piperidin-3-yl)-N-(quinolin-4-ylmethyl)benzamide
2-{3-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
N-[(2R,3R)-1'-[(4-hydroxy-3-methoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
3-[2-(methylsulfanyl)benzoyl]-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
N,1,3-trimethyl-N-(thian-4-yl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-{5-[1-(thian-4-yl)pyrrolidin-2-yl]thiophene-2-carbonyl}piperidin-4-ol
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2,6-dimethylquinoline-4-carboxamide
4-{[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]sulfamoyl}-N-(propan-2-yl)benzamide
1-[4-(benzyloxy)piperidin-1-yl]-3-(3-chloro-1H-1,2,4-triazol-5-yl)propan-1-one
2-methanesulfonamido-N-[(3R,4S)-4-propyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]acetamide
ethyl 5-[({[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]carbamoyl}amino)methyl]furan-2-carboxylate
1-{2-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-3,3-dimethylurea
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide