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1-({1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
N-[(6-hydroxypyrimidin-4-yl)methyl]-4-(piperidin-1-yl)butanamide
1-(4-chlorophenyl)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]cyclobutane-1-carboxamide
N-cyclopentyl-2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)acetamide
9-[3-(dimethylamino)-1,2,4-thiadiazol-5-yl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
N-{2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}acetamide
2-{1-[(1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-2-amine
N-[2-(7-{[2-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxane-4-carboxamide
3,5-dimethoxy-2-({methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)benzoic acid
5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-N-[1-(pyrimidin-4-yl)ethyl]pyridin-2-amine
N-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[(4-acetamidophenyl)methyl]-2-[4-(hydroxymethyl)piperidin-1-yl]acetamide
4-ethyl-3-{1-[(5-fluoro-2-methoxyphenyl)methyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S)-N-ethyl-1-(1H-imidazol-2-ylmethyl)-4-[3-(3-methyl-1H-pyrazol-1-yl)propanamido]pyrrolidine-2-carboxamide
1-(3-{[5-methyl-6-(piperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}propanamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
(4aR,7aS)-1-acetyl-4-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cyclopentyl-N-(2-methylprop-2-en-1-yl)-6-oxopiperidine-3-carboxamide
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[(2E)-2-methylbut-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-2-{5-[(2-phenylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-imidazole
3-{[1-({4-[1-(dimethylamino)ethyl]phenyl}methyl)piperidin-4-yl]methyl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2-methoxyethyl)-8-[2-methyl-2-(1H-pyrrol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidine-3-carbonyl]pyridine
(3E)-1-[(3S,4S)-3-hydroxy-4-[4-(pyridin-2-ylmethyl)piperazin-1-yl]pyrrolidin-1-yl]hex-3-en-1-one
(1S,5R)-6-benzyl-3-(2-chlorobenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
4-{3-[2-(4-fluorophenyl)azetidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(furan-2-ylmethyl)amine
N-(1-benzylpyrrolidin-3-yl)-3-[1-(3-phenylpropyl)piperidin-4-yl]propanamide
methyl 3-[(3S,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoate
N-[(2-methoxyphenyl)methyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-(prop-2-en-1-yl)acetamide
8-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
8-(2-amino-6-methylpyrimidin-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-phenylpiperidin-4-ol
3-methyl-7-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-[(2-fluorophenyl)methyl]-N-[3-(methylsulfanyl)propyl]-6-oxopiperidine-3-carboxamide
(3R,4R)-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-[2-(oxan-4-yl)ethyl]benzamide
1-ethyl-8-(1-hydroxypropan-2-yl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-ethyl-N-(pyridin-4-ylmethyl)azepane-4-carboxamide
[2-(3-methoxyphenyl)-1-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]ethyl](methyl)(pyridin-2-ylmethyl)amine
7-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-N,N,2-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-{4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}pyrazine
2-amino-5-methyl-4-(4-methyl-1,3-thiazol-2-yl)-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-(2-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
4-(1H-imidazol-1-ylmethyl)-2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazole
[(2S)-1-(3,5,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-2-yl]methanol
{1-[({[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]cyclopropyl}methanol