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N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)-1-(oxan-4-yl)piperidine-4-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]pyrimidin-4-ol
(1R,7S)-3-(4-fluoro-2-methylphenyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(2-methylprop-2-en-1-yl)-1,3-oxazole-4-carboxamide
1-[2-(dimethylamino)ethyl]-4-ethyl-3-[1-(oxane-4-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
4-(1-benzyl-5-methyl-1H-1,2,3-triazole-4-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
N-[(1S,2R)-2-[(1-acetylpiperidin-4-yl)amino]cyclobutyl]-4-(1H-imidazol-1-yl)benzamide
1-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-(2-methoxyethyl)-N-[(3-methoxyphenyl)methyl]-3,5-dimethyl-1H-indole-2-carboxamide
3-(benzenesulfonyl)-1-(6-hydroxy-4-methyl-1,4-diazepan-1-yl)propan-1-one
1-[2-(dimethylamino)-4-({2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4-(5-amino-1H-pyrazole-3-carbonyl)-5-methyl-1-(3-methylphenyl)piperazin-2-one
2-amino-4-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
2-[4-(1-benzofuran-2-ylmethyl)morpholin-3-yl]-N-(1H-indazol-5-yl)acetamide
2-[(3-chlorophenyl)methyl]-N-(1-hydroxy-2-methylpropan-2-yl)-1,3-benzoxazole-6-carboxamide
4-[1-(2,3-dihydro-1H-inden-2-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-N-methylpyridin-2-amine
N-{4-oxo-4-[2-oxo-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]butyl}acetamide
2-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]benzonitrile
N-cyclohexyl-3-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]propanamide
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
2,6-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]quinoline-4-carboxamide
3-{[2-(ethanesulfonyl)ethyl]sulfamoyl}-N-ethyl-N-methylbenzamide
(4aS,8aR)-6-[(2-methylphenyl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
7-(6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-2H-1-benzopyran-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-[2-(2-chlorophenyl)ethyl]-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methoxybenzamide
N-methyl-5-(propan-2-yl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-(cyclopropylmethyl)-5-(2,2-dimethyloxane-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(1S,6R)-3-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-(2-{7-[(3,5-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
N-[3-(4-methoxyphenyl)propyl]-6-[(3R)-3-methylpiperazin-1-yl]pyridine-3-carboxamide
N-(6-phenoxypyridin-3-yl)-1-[3-(1H-pyrazol-4-yl)propanoyl]piperidine-4-carboxamide
5,8-dimethoxy-2-(3-methylphenyl)-3-(morpholin-4-ylmethyl)quinoline
1-methyl-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}-1H-1,3-benzodiazole-5-carboxamide
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
N-(4-fluorophenyl)-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-amine
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
N-(2H-1,3-benzodioxol-5-yl)-1-[(3,7-dimethyl-1H-indol-2-yl)methyl]piperidin-3-amine
2-(propan-2-yl)-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2,5-dihydro-1H-pyrrole
1-methyl-1'-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(4H-1,2,4-triazol-4-yl)propan-1-one
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]acetamide
2-{[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-5-ethyl-1,3,4-oxadiazole
2-(3-hydroxypropyl)-9-[(2R)-5-oxopyrrolidine-2-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
5-{3-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-3-oxopropyl}imidazolidine-2,4-dione
1-(cyclohexylmethyl)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-6-oxopiperidine-3-carboxamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine