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{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amine
5-(3-fluorophenoxymethyl)-N-[5-oxo-1-(propan-2-yl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
2-(6-methoxynaphthalen-2-yl)-4-(1H-pyrrole-2-carbonyl)morpholine
4-[(6-chloroquinolin-2-yl)methyl]-N,N-dimethylpiperazine-1-sulfonamide
1-(furan-2-ylmethyl)-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-3-carboxamide
3-(3-fluorophenyl)-N-[(4-methyl-5-oxomorpholin-2-yl)methyl]benzamide
3-[3-cyclopropyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]quinoline
1-(4-hydroxy-4-methylazepan-1-yl)-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
N-butyl-4-{[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
N1-(4-ethyl-5-methylpyrimidin-2-yl)pentane-1,5-diamine
ethyl 4-{3-[(3-methoxyphenyl)methyl]-1,2-oxazole-5-amido}piperidine-1-carboxylate
N-(1-phenylethyl)-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2-[5-methyl-4-(4-phenylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
3,3,3-trifluoro-1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]propan-1-one
N-(4-methylphenyl)-2-({2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}amino)propanamide
N-(1-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-2-carboxamide
N-(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
5-(methoxymethyl)-N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}furan-2-carboxamide
1-benzyl-3-(2-methoxyethyl)-8-{[4-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
1-ethyl-4-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carbonyl)piperazine
methyl 1-[(3R,5S)-1-{[5-(2-chlorophenyl)furan-2-yl]methyl}-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-phenyl-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carboxamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-chloro-5-acetamido-N-[1-(4-methylpyridin-2-yl)propyl]benzamide
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-[2-(methylsulfanyl)ethyl]piperazine
{2-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-8-methylquinolin-3-yl}methanol
2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carboxylic acid
3-{3-[cyclohexyl(methyl)amino]propyl}-8-(furan-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(pyrazine-2-carbonyl)-1,4-diazepan-6-ol
6-(2,5-dimethylfuran-3-yl)-7-(prop-2-en-1-yl)-2-(thiomorpholine-4-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
4-{[(2S,5R)-5-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)oxolan-2-yl]methyl}benzonitrile
2-acetyl-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]benzamide
1,4,6-trimethyl-3-[2-(4-methylpentyl)morpholine-4-carbonyl]-1,2-dihydropyridin-2-one
2-(2-methoxyethyl)-1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-4-methyl-1,2,3-thiadiazole-5-carboxamide
3-(3,4-difluorophenyl)-5-[2-(1H-pyrazol-1-yl)ethyl]-1,2,4-oxadiazole
(2S,4R)-4-amino-N-methyl-1-{5-[(phenylsulfanyl)methyl]furan-2-carbonyl}pyrrolidine-2-carboxamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-[1-(thiophen-2-yl)ethyl]piperidine-3-carboxamide
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1H-1,2,4-triazol-3-ylsulfanyl)ethan-1-one
N-benzyl-N-(2-hydroxyethyl)-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidine
(2R,3R,6R)-5-(1H-indole-6-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-methyl-8-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}ethan-1-one
N-ethyl-5-(3-methoxyphenoxymethyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
3-{2-[ethyl({[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amino]-1-hydroxyethyl}phenol
8-(2,5-dimethylfuran-3-carbonyl)-2-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one